Browsing by Author Luque Garriga, F. Xavier

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Issue DateTitleAuthor(s)
12-Feb-20141,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: synthesis, pharmacological evaluation and mechanistic studiesDi Pietro, O.; Viayna, Elisabet; Vicente García, Esther; Bartolini, Manuela; Ramón, Rosario; Juárez-Jiménez, Jordi; Clos, Victòria; Pérez Fernández, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego
9-Feb-2024Acetylcholinesterase: A versatile template to coin potent modulators of multiple therapeutic targetsLuque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
24-Feb-2015Activitats per a l'alumnat de secundària "Farmaestiu"Bidon-Chanal Badia, Axel; Juárez, Jordi; Luque Garriga, F. Xavier; Amat, Concepció; Saldaña-Ruíz, Sandra; Miquel Colomé, Jordi; García Montoya, Encarna; Badía Palacín, Josefa; Escolano Mirón, Carmen; Esteva de Sagrera, Juan, 1948-; Muñoz-Torrero López-Ibarra, Diego; Pallàs i Llibería, Mercè, 1964-; Miñarro Carmona, Montserrat; Plou, Silvina
5-Mar-2021Azobioisosteres of Curcumin with Pronounced Activity against Amyloid Aggregation, Intracellular Oxidative Stress, and NeuroinflammationHofmann, Julian; Ginex, Tiziana; Espargaró Colomé, Alba; Scheiner, Matthias; Gunesch, Sandra; Aragó, Marc; Stigloher, Christian; Sabaté Lagunas, Raimon; Luque Garriga, F. Xavier; Decker, Michael
19-Mar-2020Bicyclic alfa-iminophosphonates as high affinity imidazoline I2 receptor ligands for Alzheimer's diseaseAbás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Pérez, Belén; Molins i Grau, Elies; Luque Garriga, F. Xavier; Pérez Lozano, Pilar; Jonghe, Steven de; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, María Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Pallàs i Llibería, Mercè, 1964-; Callado, Luis F.; Escolano Mirón, Carmen
5-May-2017Breakthroughs in Medicinal Chemistry: New targets and mechanisms, new drugs, new hopesMuñoz-Torrero López-Ibarra, Diego; Mangoni, Arduino A.; Guillou, Catherine; Collina, Simona; Vanden Eynde, Jean Jacques; Rautio, Jarkko; Keseru, György M.; Hulme, Christopher; Chibale, Kelly; Luque Garriga, F. Xavier; Karaman, Rafik; Gütschow, Michael; Liu, Hong; Ragno, Rino
2018Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-2Muñoz-Torrero López-Ibarra, Diego; Mangoni, Arduino A.; Liu, Hong; Hulme, Christopher; Rautio, Jarkko; Karaman, Rafik; Sousa, Maria Emília de; Prokai-Tatrai, Katalin; Sabatier, Jean-Marc; Siciliano, Carlo; Luque Garriga, F. Xavier; Kokotos, George; Ragno, Rino; Collina, Simona; Guillou, Catherine; Gütschow, Michael; Agrofoglio, Luigi A.
2019Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-4Mangoni, Arduino A.; Guillou, Catherine; Vanden Eynde, Jean Jacques; Hulme, Christopher; Jampilek, Josef; Li, Wei; Prokai-Tatrai, Katalin; Rautio, Jarkko; Collina, Simona; Tuccinardi, Tiziano; Sousa, Maria Emília de; Sabatier, Jean-Marc; Galdiero, Stefania; Karaman, Rafik; Kokotos, George; Torri, Giangiacomo; Luque Garriga, F. Xavier; Vasconcelos, M. Helena; Hadjipavlou-Litina, Dimitra; Siciliano, Carlo; Gütschow, Michael; Ragno, Rino; Gomes, Paula A. C; Agrofoglio, Luigi A.; Muñoz-Torrero López-Ibarra, Diego
2019Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-5Mangoni, Arduino A.; Vanden Eynde, Jean Jacques; Jampilek, Josef; Hadjipavlou-Litina, Dimitra; Liu, Hong; Reynisson, Jóhannes; Sousa, Maria Emília de; Gomes, Paula A. C; Prokai-Tatrai, Katalin; Tuccinardi, Tiziano; Sabatier, Jean-Marc; Luque Garriga, F. Xavier; Rautio, Jarkko; Karaman, Rafik; Vasconcelos, M. Helena; Gemma, Sandra; Galdiero, Stefania; Hulme, Christopher; Collina, Simona; Gütschow, Michael; Kokotos, George; Siciliano, Carlo; Capasso, Raffaele; Agrofoglio, Luigi A.; Ragno, Rino; Muñoz-Torrero López-Ibarra, Diego
28-Dec-2019Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6Vanden Eynde, Jean Jacques; Mangoni, Arduino A.; Rautio, Jarkko; Leprince, Jérôme; Azuma, Yasu-Taka; García-Sosa, Alfonso T.; Hulme, Christopher; Jampilek, Josef; Karaman, Rafik; Li, Wei; Gomes, Paula A. C; Hadjipavlou-Litina, Dimitra; Capasso, Raffaele; Geronikaki, Athina; Cerchia, Laura; Sabatier, Jean-Marc; Ragno, Rino; Tuccinardi, Tiziano; Trabocchi, Andrea; Winum, Jean-Yves; Luque Garriga, F. Xavier; Prokai-Tatrai, Katalin; Spetea, Mariana; Gütschow, Michael; Kosalec, Ivan; Guillou, Catherine; Vasconcelos, M. Helena; Kokotos, George; Rastelli, Giulio; de Sousa, Maria Emília; Manera, Clementina; Gemma, Sandra; Mangani, Stefano; Siciliano, Carlo; Galdiero, Stefania; Liu, Hong; Scott, Peter J. H.; de los Ríos, Cristóbal; Agrofoglio, Luigi A.; Collina, Simona; Guedes, Rita C.; Muñoz-Torrero López-Ibarra, Diego
4-Jan-2013CO rebinding kinetics and molecular dynamics simulations highlight dynamic regulation of internal cavities in human cytoglobinGabba, Matteo; Abbruzzetti, Stefania; Spyrakis, Francesca; Forti, Flavio; Bruno, Stefano; Mozzarelli, Andrea; Luque Garriga, F. Xavier; Viappiani, Cristiano; Cozzini, Pietro; Nardini, Marco; Germani, Francesca; Bolognesi, Martino; Moens, Luc; Dewilde, Sylvia
6-Nov-2004Conjugate Addition to Phenylglycinol-Derived Unsaturated ä-Lactams. Enantioselective Synthesos of Uleine AlkaloidsAmat Tusón, Mercedes; Pérez Bosch, Maria; Llor Brunés, Núria; Escolano Mirón, Carmen; Luque Garriga, F. Xavier; Molins i Grau, Elies; Bosch Cartes, Joan
19-Jul-2019Desarrollos metodológicos en la exploración de la especie bioactiva en fármacos: Búsqueda de agentes antimaláricosViayna Gaza, Antonio
30-Jul-2018Determination of the protonation preferences of bilin pigments in cryptophyte antenna complexesCorbella Morató, Marina; Toa, Zi. S. D.; Scholes, Gregory D.; Luque Garriga, F. Xavier; Curutchet Barat, Carles E.
21-Feb-2019Development of a Structure-Based, pH-Dependent Lipophilicity Scale of Amino Acids from Continuum Solvation CalculationsZamora Ramírez, William J.; Campanera Alsina, Josep Maria; Luque Garriga, F. Xavier
11-Mar-2020Dioxygen Binding and Sensing ProteinsEstrín, Darío; Luque Garriga, F. Xavier; Ilangovan, Govindasamy; Zweier, Jay L
4-May-2012Disseny, síntesi, avaluació farmacològica i modelatge molecular de nous inhibidors de l’acetilcolinesterasa de lloc d’unió dualGaldeano Cantador, Carlos
18-Jul-2018Electrostatic tuning of the ligand binding mechanism by Glu27 in nitrophorin 7Abbruzzetti, Stefania; Allegri, Alessandro; Bidon-Chanal Badia, Axel; Ogata, Hideaki; Soavi, Giancarlo; Cerullo, Giulio; Bruno, Stefano; Montali, Chiara; Luque Garriga, F. Xavier; Viappiani, Cristiano
5-Nov-2021Elucidating the activation mechanism of AMPK by direct pan-activator PF-739Aledavood, Elnaz; Gheeraert, Aria; Forte, Alessia; Vuillon, Laurent; Rivalta, Ivan; Luque Garriga, F. Xavier; Estarellas, Carolina
4-Aug-2017Enantioselective Synthesis of Spiro[indolizidine-1,3 '-oxindoles]Pérez Bosch, Maria; Ramos, Carlos; Massi, Lucia; Gazzola, Silvia; Taglienti, Chiara; Yayik, Nihan; Molins i Grau, Elies; Viayna Gaza, Antonio; Luque Garriga, F. Xavier; Bosch Cartes, Joan; Amat Tusón, Mercedes