Search
Add filters:
Use filters to refine the search results.
Results 1-10 of 10 (Search time: 0.009 seconds).
- previous
- 1
- next
Item hits:
Issue Date | Title | Author(s) |
---|---|---|
12-Feb-2014 | 1,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: synthesis, pharmacological evaluation and mechanistic studies | Di Pietro, O.; Viayna, Elisabet; Vicente García, Esther; Bartolini, Manuela; Ramón, Rosario; Juárez-Jiménez, Jordi; Clos, Victòria; Pérez Fernández, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego |
27-Mar-2014 | Synthesis and multi-target biological profiling of a novel family of rhein derivatives as disease-modifying anti-Alzheimer agents | Viayna, Elisabet; Sola, Irene; Bartolini, Manuela; De Simone, Angela; Tapia-Rojas, Cheril; Serrano, Felipe G.; Sabaté Lagunas, Raimon; Juárez-Jiménez, Jordi; Pérez Fernández, Belén; Luque Garriga, F. Xavier; Andrisano, Vincenza; Clos, Victòria; Inestrosa, Nibaldo C.; Muñoz-Torrero López-Ibarra, Diego |
1-Oct-2014 | Shogaol-huprine hybrids: Dual antioxidant and anticholinesterase agents with beta-amyloid and tau anti-aggregating properties | Pérez Areales, Francisco Javier; Di Pietro, O.; Espargaró Colomé, Alba; Vallverdú i Queralt, Anna; Galdeano Cantador, Carlos; Ragusa, Ilaria M.; Viayna, Elisabet; Guillou, Catherine; Clos, Victòria; Pérez Fernández, Belén; Sabaté Lagunas, Raimon; Lamuela Raventós, Rosa Ma.; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
12-Sep-2014 | Tetrahydrobenzo[h][1,6]naphthyridine-6-chlorotacrine hybrids as a new family of anti-Alzheimer agents targeting beta-amyloid, tau, and cholinesterase pathologies | Di Pietro, O.; Pérez Areales, Francisco Javier; Juárez-Jiménez, Jordi; Espargaró Colomé, Alba; Clos, Victòria; Pérez Fernández, Belén; Lavilla Grífols, Rodolfo; Sabaté Lagunas, Raimon; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
5-May-2017 | Breakthroughs in Medicinal Chemistry: New targets and mechanisms, new drugs, new hopes | Muñoz-Torrero López-Ibarra, Diego; Mangoni, Arduino A.; Guillou, Catherine; Collina, Simona; Vanden Eynde, Jean Jacques; Rautio, Jarkko; Keseru, György M.; Hulme, Christopher; Chibale, Kelly; Luque Garriga, F. Xavier; Karaman, Rafik; Gütschow, Michael; Liu, Hong; Ragno, Rino |
2018 | Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-2 | Muñoz-Torrero López-Ibarra, Diego; Mangoni, Arduino A.; Liu, Hong; Hulme, Christopher; Rautio, Jarkko; Karaman, Rafik; Sousa, Maria Emília de; Prokai-Tatrai, Katalin; Sabatier, Jean-Marc; Siciliano, Carlo; Luque Garriga, F. Xavier; Kokotos, George; Ragno, Rino; Collina, Simona; Guillou, Catherine; Gütschow, Michael; Agrofoglio, Luigi A. |
15-May-2017 | Unveiling a Novel Transient Druggable Pocket in BACE-1 through Molecular Simulations: Conformational Analysis and Binding Mode of Multisite Inhibitors | Di Pietro, O.; Juárez Jiménez, Jordi; Muñoz-Torrero López-Ibarra, Diego; Laughton, Charles A.; Luque Garriga, F. Xavier |
2019 | Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-4 | Mangoni, Arduino A.; Guillou, Catherine; Vanden Eynde, Jean Jacques; Hulme, Christopher; Jampilek, Josef; Li, Wei; Prokai-Tatrai, Katalin; Rautio, Jarkko; Collina, Simona; Tuccinardi, Tiziano; Sousa, Maria Emília de; Sabatier, Jean-Marc; Galdiero, Stefania; Karaman, Rafik; Kokotos, George; Torri, Giangiacomo; Luque Garriga, F. Xavier; Vasconcelos, M. Helena; Hadjipavlou-Litina, Dimitra; Siciliano, Carlo; Gütschow, Michael; Ragno, Rino; Gomes, Paula A. C; Agrofoglio, Luigi A.; Muñoz-Torrero López-Ibarra, Diego |
14-Aug-2019 | Synthesis, in vitro profiling, and in vivo efficacy studies of a new family of multitarget anti-Alzheimer compounds | Pérez Areales, Francisco Javier; Garrido, María; Aso Pérez, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró Colomé, Alba; Ginex, Tiziana; Sabaté Lagunas, Raimon; Pérez, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Ferrer, Isidro (Ferrer Abizanda); Ciruela Alférez, Francisco; Messeguer i Peypoch, Àngel, 1946-; Muñoz-Torrero López-Ibarra, Diego |
28-Dec-2019 | Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6 | Vanden Eynde, Jean Jacques; Mangoni, Arduino A.; Rautio, Jarkko; Leprince, Jérôme; Azuma, Yasu-Taka; García-Sosa, Alfonso T.; Hulme, Christopher; Jampilek, Josef; Karaman, Rafik; Li, Wei; Gomes, Paula A. C; Hadjipavlou-Litina, Dimitra; Capasso, Raffaele; Geronikaki, Athina; Cerchia, Laura; Sabatier, Jean-Marc; Ragno, Rino; Tuccinardi, Tiziano; Trabocchi, Andrea; Winum, Jean-Yves; Luque Garriga, F. Xavier; Prokai-Tatrai, Katalin; Spetea, Mariana; Gütschow, Michael; Kosalec, Ivan; Guillou, Catherine; Vasconcelos, M. Helena; Kokotos, George; Rastelli, Giulio; de Sousa, Maria Emília; Manera, Clementina; Gemma, Sandra; Mangani, Stefano; Siciliano, Carlo; Galdiero, Stefania; Liu, Hong; Scott, Peter J. H.; de los Ríos, Cristóbal; Agrofoglio, Luigi A.; Collina, Simona; Guedes, Rita C.; Muñoz-Torrero López-Ibarra, Diego |
Discover
Subject