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Issue Date | Title | Author(s) |
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12-Feb-2014 | 1,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: synthesis, pharmacological evaluation and mechanistic studies | Di Pietro, O.; Viayna, Elisabet; Vicente García, Esther; Bartolini, Manuela; Ramón, Rosario; Juárez-Jiménez, Jordi; Clos, Victòria; Pérez Fernández, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego |
27-Mar-2014 | Synthesis and multi-target biological profiling of a novel family of rhein derivatives as disease-modifying anti-Alzheimer agents | Viayna, Elisabet; Sola, Irene; Bartolini, Manuela; De Simone, Angela; Tapia-Rojas, Cheril; Serrano, Felipe G.; Sabaté Lagunas, Raimon; Juárez-Jiménez, Jordi; Pérez Fernández, Belén; Luque Garriga, F. Xavier; Andrisano, Vincenza; Clos, Victòria; Inestrosa, Nibaldo C.; Muñoz-Torrero López-Ibarra, Diego |
1-Oct-2014 | Shogaol-huprine hybrids: Dual antioxidant and anticholinesterase agents with beta-amyloid and tau anti-aggregating properties | Pérez Areales, Francisco Javier; Di Pietro, O.; Espargaró Colomé, Alba; Vallverdú i Queralt, Anna; Galdeano Cantador, Carlos; Ragusa, Ilaria M.; Viayna, Elisabet; Guillou, Catherine; Clos, Victòria; Pérez Fernández, Belén; Sabaté Lagunas, Raimon; Lamuela Raventós, Rosa Ma.; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
12-Sep-2014 | Tetrahydrobenzo[h][1,6]naphthyridine-6-chlorotacrine hybrids as a new family of anti-Alzheimer agents targeting beta-amyloid, tau, and cholinesterase pathologies | Di Pietro, O.; Pérez Areales, Francisco Javier; Juárez-Jiménez, Jordi; Espargaró Colomé, Alba; Clos, Victòria; Pérez Fernández, Belén; Lavilla Grífols, Rodolfo; Sabaté Lagunas, Raimon; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
14-Sep-2015 | Stereocontrolled annulations of indolo[2,3-a]quinolizidine-derived lactams with a silylated Nazarov reagent. Access to allo and epiallo yohimbine-type derivatives | Arioli, Federica; Pérez Bosch, Maria; Are, Celeste; Estarellas, Carolina; Luque Garriga, F. Xavier; Bosch Cartes, Joan; Amat Tusón, Mercedes |
8-Nov-2012 | Role of PheE15 gate in ligand entry and nitric oxide detoxification function of Mycobacterium tuberculosis truncated hemoglobin N | Oliveira, Ana; Singh, Sandeep; Bidon-Chanal Badia, Axel; Forti, Flavio; Martí, Marcelo A.; Boechi, Leonardo; Estrín, Darío; Dikshit, Kanak L.; Luque Garriga, F. Xavier |
13-Nov-2015 | Interaction of the N-(3-Methylpyridin-2-yl)amide Derivatives of Flurbiprofen and Ibuprofen with FAAH: Enantiomeric Selectivity and Binding Mode | Karlsson, Jessica; Morgillo, Carmine Marco; Deplano, Alessandro; Smaldone, Giovanni; Pedone, Emilia; Luque Garriga, F. Xavier; Svensson, Mona; Novellino, Ettore; Congiu, Cenzo; Onnis, Valentina; Catalanotti, Bruno; Fowler, Christopher J. |
5-May-2017 | Breakthroughs in Medicinal Chemistry: New targets and mechanisms, new drugs, new hopes | Muñoz-Torrero López-Ibarra, Diego; Mangoni, Arduino A.; Guillou, Catherine; Collina, Simona; Vanden Eynde, Jean Jacques; Rautio, Jarkko; Keseru, György M.; Hulme, Christopher; Chibale, Kelly; Luque Garriga, F. Xavier; Karaman, Rafik; Gütschow, Michael; Liu, Hong; Ragno, Rino |
14-Apr-2015 | New polycyclic dual inhibitors of the wild type and the V27A mutant M2 channel of the influenza A virus with unexpected binding mode | Rey Carrizo, Matías; Gazzarrini, Sabrina; Llabrés Prat, Salomé; Frigolé Vivas, Marta; Juárez Jiménez, Jordi; Font Bardia, Ma. Mercedes; Naesens, Lieve; Moroni, Anna; Luque Garriga, F. Xavier; Vázquez Cruz, Santiago |
12-Jun-2021 | New trimethoprim-like molecules: bacteriological evaluation and insights into their action | Jorba, Marta; Pedrola, Marina; Ghashghaei, Ouldouz; Herráez, Rocío; Campos Vicens, Lluís; Luque Garriga, F. Xavier; Lavilla Grífols, Rodolfo; Viñas, Miquel |
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