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Issue DateTitleAuthor(s)
12-Feb-20141,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: synthesis, pharmacological evaluation and mechanistic studiesDi Pietro, O.; Viayna, Elisabet; Vicente García, Esther; Bartolini, Manuela; Ramón, Rosario; Juárez-Jiménez, Jordi; Clos, Victòria; Pérez Fernández, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego
1-Aug-2013Dual inhibitors of beta-amyloid aggregation and acetylcholinesterase as multi-target anti-Alzheimer drug candidatesViayna, Elisabet; Sabaté Lagunas, Raimon; Muñoz-Torrero López-Ibarra, Diego
27-Mar-2014Synthesis and multi-target biological profiling of a novel family of rhein derivatives as disease-modifying anti-Alzheimer agentsViayna, Elisabet; Sola, Irene; Bartolini, Manuela; De Simone, Angela; Tapia-Rojas, Cheril; Serrano, Felipe G.; Sabaté Lagunas, Raimon; Juárez-Jiménez, Jordi; Pérez Fernández, Belén; Luque Garriga, F. Xavier; Andrisano, Vincenza; Clos, Victòria; Inestrosa, Nibaldo C.; Muñoz-Torrero López-Ibarra, Diego
1-Oct-2014Shogaol-huprine hybrids: Dual antioxidant and anticholinesterase agents with beta-amyloid and tau anti-aggregating propertiesPérez Areales, Francisco Javier; Di Pietro, O.; Espargaró Colomé, Alba; Vallverdú i Queralt, Anna; Galdeano Cantador, Carlos; Ragusa, Ilaria M.; Viayna, Elisabet; Guillou, Catherine; Clos, Victòria; Pérez Fernández, Belén; Sabaté Lagunas, Raimon; Lamuela Raventós, Rosa Ma.; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
12-Sep-2014Tetrahydrobenzo[h][1,6]naphthyridine-6-chlorotacrine hybrids as a new family of anti-Alzheimer agents targeting beta-amyloid, tau, and cholinesterase pathologiesDi Pietro, O.; Pérez Areales, Francisco Javier; Juárez-Jiménez, Jordi; Espargaró Colomé, Alba; Clos, Victòria; Pérez Fernández, Belén; Lavilla Grífols, Rodolfo; Sabaté Lagunas, Raimon; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
Mar-2014Thioflavin-S staining of bacterial inclusion bodies for the fast, simple, and inexpensive screening of amyloid aggregation inhibitorsPouplana, Sergi; Espargaró Colomé, Alba; Galdeano Cantador, Carlos; Viayna, Elisabet; Sola, Irene; Ventura, Salvador; Muñoz-Torrero López-Ibarra, Diego; Sabaté Lagunas, Raimon
10-Mar-2015Multigram synthesis and in vivo efficacy studies of a novel multitarget anti-Alzheimer's compoundSola, Irene; Viayna, Elisabet; Gómez Nadal, Tània; Galdeano Cantador, Carlos; Cassina, Matteo; Camps García, Pelayo; Romeo, Margherita; Diomede, Luisa; Salmona, Mario; Franco, Pilar; Schaeffer, Mireille; Colantuono, Diego; Robin, David; Brunner, Daniela; Taub, Nicole; Hutter-Paier, Birgit; Muñoz-Torrero López-Ibarra, Diego
22-Mar-2016Ultra rapid in vivo screening for anti-Alzheimer anti-amyloid drugsEspargaró Colomé, Alba; Medina, Aina; Di Pietro, O.; Muñoz-Torrero López-Ibarra, Diego; Sabaté Lagunas, Raimon
2018Development of hybrid compounds to tackle Alzheimer’s diseaseMuñoz-Torrero López-Ibarra, Diego; Pérez Areales, Francisco Javier
2021Clock/Sleep-Dependent Learning and Memory in Male 3xTg-AD Mice at Advanced Disease Stages and Extrinsic Effects of Huprine X and the Novel Multitarget Agent AVCRI104P3Giménez Llort, Lydia; Santana-Santana, Mikel; Ratia, Míriam; Pérez, Belén; Camps García, Pelayo; Muñoz-Torrero López-Ibarra, Diego; Badía, A. (Albert); Clos, Victòria