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Issue DateTitleAuthor(s)
30-Oct-2022Three to Tango: Inhibitory Effect of Quercetin and Apigenin on Acetylcholinesterase, Amyloid-β Aggregation and Acetylcholinesterase-Amyloid InteractionAlvarez-Berbel, Irene; Espargaró Colomé, Alba; Viayna, Elisabet; Caballero Hernández, Ana Belén; Busquets i Viñas, Ma. Antonia; Gámez Enamorado, Patrick; Luque Garriga, F. Xavier; Sabaté Lagunas, Raimon
27-May-2022Design, synthesis, and in vitro, in silico and in cellulo evaluation of new pyrimidine and pyridine amide and carbamate derivatives as multi-functional cholinesterase inhibitorsBortolami, Martina; Pandolfi, Fabiana; Tudino, Valeria; Messore, Antonella; Madia, Valentina Noemi; De Vita, Daniela; Di Santo, Roberto; Costi, Roberta; Romeo, Isabella; Alcaro, Stefano; Colone, Marisa; Stringaro, Annarita; Espargaró Colomé, Alba; Sabaté Lagunas, Raimon; Scipione, Luigi
11-Jan-2023New cyclopentaquinoline and 3,5-dichlorobenzoic acid hybrids with neuroprotection against oxidative stress for the treatment of Alzheimer's diseaseCzarnecka, Kamila; Malgorzata, Girek; Krecisz, Pawel; Skibinski, Robert; Latka, Kamil; Jonczyk, Jakub; Bajda, Marek; Szymczyk, Piotr; Galita, Grzegorz; Kabzinski, Jacek; Majesterek, Ireneusz; Espargaró Colomé, Alba; Sabaté Lagunas, Raimon; Szymanski, Pawel
7-Dec-2020Pharmacophore Modeling and 3D-QSAR Study of Indole and Isatin Derivatives as Antiamyloidogenic Agents Targeting Alzheimer's DiseasePurgatorio, Rosario; Gambacorta, Nicola; Catto, Marco; de Candia, Modesto; Pisani, Leonardo; Espargaró Colomé, Alba; Sabaté Lagunas, Raimon; Cellamare, Saverio; Nicolotti, Orazio; Altomare, Cosimo D.
2021From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effectsPont Masanet, Caterina; Ginex, Tiziana; Griñán Ferré, Christian; Scheiner, Matthias; Mattellone, Alexia; Martínez, Noemí; Arce, Elsa M.; Soriano-Fernández, Yolanda; Naldi, Marina; De Simone, Angela; Barenys Espadaler, Marta; Gómez Catalán, Jesús; Pérez, Belén; Sabaté Lagunas, Raimon; Andrisano, Vincenza; Loza, María Isabel; Brea, José; Bartolini, Manuela; Bolognesi, Maria Laura; Decker, Michael; Pallàs i Llibería, Mercè, 1964-; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
2022Anti-Amyloid Drug Screening Methods Using Bacterial Inclusion BodiesCaballero Hernández, Ana Belén; Gámez Enamorado, Patrick; Sabaté Lagunas, Raimon; Espargaró Colomé, Alba