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Results 1-10 of 18 (Search time: 0.025 seconds).
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Issue DateTitleAuthor(s)
12-Feb-20141,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: synthesis, pharmacological evaluation and mechanistic studiesDi Pietro, O.; Viayna, Elisabet; Vicente García, Esther; Bartolini, Manuela; Ramón, Rosario; Juárez-Jiménez, Jordi; Clos, Victòria; Pérez Fernández, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego
27-Mar-2014Synthesis and multi-target biological profiling of a novel family of rhein derivatives as disease-modifying anti-Alzheimer agentsViayna, Elisabet; Sola, Irene; Bartolini, Manuela; De Simone, Angela; Tapia-Rojas, Cheril; Serrano, Felipe G.; Sabaté Lagunas, Raimon; Juárez-Jiménez, Jordi; Pérez Fernández, Belén; Luque Garriga, F. Xavier; Andrisano, Vincenza; Clos, Victòria; Inestrosa, Nibaldo C.; Muñoz-Torrero López-Ibarra, Diego
10-Apr-2014rDock: A Fast, Versatile and Open Source Program for Docking Ligands to Proteins and Nucleic AcidsRuiz Carmona, Sergio; Alvarez-Garcia, Daniel; Foloppe, Nicolas; Garmendia-Doval, A. Beatriz; Juhos, Szilveszter; Schmidtke, Peter; Barril Alonso, Xavier; Hubbard, Roderick E.; Morley, S. David
1-Oct-2014Shogaol-huprine hybrids: Dual antioxidant and anticholinesterase agents with beta-amyloid and tau anti-aggregating propertiesPérez Areales, Francisco Javier; Di Pietro, O.; Espargaró Colomé, Alba; Vallverdú i Queralt, Anna; Galdeano Cantador, Carlos; Ragusa, Ilaria M.; Viayna, Elisabet; Guillou, Catherine; Clos, Victòria; Pérez Fernández, Belén; Sabaté Lagunas, Raimon; Lamuela Raventós, Rosa Ma.; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
12-Sep-2014Tetrahydrobenzo[h][1,6]naphthyridine-6-chlorotacrine hybrids as a new family of anti-Alzheimer agents targeting beta-amyloid, tau, and cholinesterase pathologiesDi Pietro, O.; Pérez Areales, Francisco Javier; Juárez-Jiménez, Jordi; Espargaró Colomé, Alba; Clos, Victòria; Pérez Fernández, Belén; Lavilla Grífols, Rodolfo; Sabaté Lagunas, Raimon; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
22-Mar-2016Ultra rapid in vivo screening for anti-Alzheimer anti-amyloid drugsEspargaró Colomé, Alba; Medina, Aina; Di Pietro, O.; Muñoz-Torrero López-Ibarra, Diego; Sabaté Lagunas, Raimon
11-Dec-2018Solvents to Fragments to Drugs: MD Applications in Drug DesignDefelipe, Lucas A.; Arcon, Juan Pablo; Modenutti, Carlos P.; Martí, Marcelo A.; Turjanski,Adrián G.; Barril Alonso, Xavier
2018PPARγ agonist-loaded PLGA-PEG nanocarriers as a potencial treatment for Alzheimer's disease: in vitro and in vivo studies.Silva Abreu, Marcelle; Calpena Campmany, Ana Cristina; Andrés Benito, Pol; Aso Pérez, Ester; Romero, Ignacio A.; Roig-Carles, David; Gromicova, Radka; Espina García, Marta; Ferrer, Isidro (Ferrer Abizanda); García, Maria Luisa; Male, David K., 1954-
24-Apr-2018The Role of SeDeM Characterizing the Active Substance and Polyvynilpyrrolidone Eliminating Metastable Forms in an Oral Lyophilizate - A Preformulation Study.Flórez Borges, Paloma; Pérez Lozano, Pilar; García Montoya, Encarna; Miñarro Carmona, Montserrat; Jo, Enric; Manich Bou, Albert; Suñé i Negre, Josep M. (Josep Maria)
29-Jun-2017Detecting similar binding pockets to enable systems polypharmacologyDuran Frigola, Miquel; Siragusa, Lydia; Ruppin, Eytan; Barril Alonso, Xavier; Cruciani, Gabriele; Aloy, Patrick, 1972-