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Title: Solid-Phase Synthesis of New Trp(Nps)-Containing Dipeptide Derivatives as TRPV1 Channel Blockers
Author: Pérez de Vega, M.J.
García-López, M.T.
Zaccaro, L.
Royo Expósito, Miriam
Albericio Palomera, Fernando
Fernández-Carvajal, A.
Ferrer-Montiel, A.
González-Muñiz, R.
Keywords: Síntesi en fase sólida
Canals iònics
Ciències de la salut
Dianes farmacològiques
Solid-phase synthesis
Ion channels
Medical sciences
Drug targeting
Issue Date: 15-Jul-2010
Publisher: MDPI Publishing
Abstract: Trp(Nps)-Lys-NH2 derivatives, bearing alkyl or guanidine groups either at the N-terminus or on the Lys side-chain or at both positions were conveniently prepared on solid-phase and evaluated as TRPV1 channel antagonists.
Note: Reproducció del document publicat a:
It is part of: Molecules, 2010, vol. 15, num. 7, p. 4924-4933
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ISSN: 1420-3049
Appears in Collections:Articles publicats en revistes (Química Inorgànica i Orgànica)

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