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Results 11-20 of 33 (Search time: 0.021 seconds).
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Issue DateTitleAuthor(s)
7-Jun-2016Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanineMartín-Gago, Pablo; Rol Rúa, Álvaro; Todorovski, Toni; Aragón Altarriba, Eric; Martin-Malpartida, Pau; Verdaguer i Espaulella, Xavier; Vallès Miret, Mariona; Fernández-Carneado, Jimena; Ponsati, Berta; Macías Hernández, María J.; Riera i Escalé, Antoni
22-Jun-2017Dialkylammonium tert-Butylmethylphosphinites: Stable Intermediates for the Synthesis of P-Stereogenic LigandsSalomó i Prat, Ernest; Prades, Amparo; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
31-Mar-2017P-Stereogenic bisphosphines with a hydrazine backbone: from N-N atropoisomerism to double nitrogen inversionPrades, Amparo; Núñez-Pertíñez, Samuel; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
2015Stereoselective synthesis of 2-acetamido-1,2-dideoxynojirimycin (DNJNAc) and ureido-DNJNAc derivatives as new hexosaminidase inhibitorsFuente Cebrián, Àlex de la; Mena-Barragán, Teresa; Farrar-Tobar, Ronald A.; Verdaguer i Espaulella, Xavier; García-Fernández, J. M.; Ortiz Mellet, Carmen; Riera i Escalé, Antoni
14-Sep-2022Design and optimization of oestrogen receptor PROTACs based on 4-hydroxytamoxifenLoren, Guillem; Espuny, Irene; Llorente Lope, Alicia; Donoghue, Craig; Verdaguer i Espaulella, Xavier; Gomis, Roger R.; Riera i Escalé, Antoni
26-Nov-2018Direct Asymmetric Hydrogenation of N-Methyl and N-Alkyl Imines with an Ir(III)H CatalystSalomó i Prat, Ernest; Gallen Ortiz, Albert; Sciortino, Giuseppe; Ujaque, Gregori; Grabulosa, Arnald; Lledós, Agustí (Lledós i Falcó); Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
20-Apr-2018P-Stereogenic and Non-P-Stereogenic Ir-MaxPHOX in the asymmetric hydrogenation of N-Aryl imines. Isolation and X-ray analysis of imine iridacyclesSalomó i Prat, Ernest; Rojo, Pep; Hernández Lladó, Pol; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
29-Dec-2014Asymmetric intermolecular cobalt-catalyzed Pauson-Khand reaction using a p-stereogenic bis-phosphaneOrgué Gassol, Sílvia; León Serrano, Thierry; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
22-Dec-2014Borane as an efficient directing group. Stereoselective 1,2-addition of organometallic reagents to borane P-stereogenic N-phosphanyliminesFlores-Gaspar, Areli; Orgué Gassol, Sílvia; Grabulosa, Arnald; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
16-Jan-2019Extending the substrate scope in the hydrogenation of unfunctionalized tetrasubstituted olefins with Ir-P stereogenic aminophosphine-oxazoline catalystsBiosca, Maria; Salomó i Prat, Ernest; Cruz Sánchez, Pol de la; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier; Pàmies, Oscar; Diéguez, Montserrat