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Issue Date | Title | Author(s) |
---|---|---|
14-Sep-2022 | Design and optimization of oestrogen receptor PROTACs based on 4-hydroxytamoxifen | Loren, Guillem; Espuny, Irene; Llorente Lope, Alicia; Donoghue, Craig; Verdaguer i Espaulella, Xavier; Gomis, Roger R.; Riera i Escalé, Antoni |
11-May-2022 | Iridium-catalyzed asymmetric hydrogenation of 2,3-diarylallyl amines with a threonine-derived P-stereogenic ligand for the synthesis of tetrahydroquinolines and tetrahydroisoquinolines | Rojo, Pep; Molinari, Medea; Cabré, Albert; García-Mateos, Clara; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier |
3-Jun-2021 | BOM-phosphinite as an electrophilic P-stereogenic transfer reagent for the synthesis of bulky phosphines. Synthesis of tert-butyl(3,5-di-tert-butylphenyl)BisP* | Rojo, Pep; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier |
12-May-2022 | Amino acids with fluorescent tetrazine ethers as bioorthogonal handles for peptide modification | Ros, Enric; Bellido, Marina; Matarin, Joan A.; Gallen, Albert; Martínez, Manuel; Rodríguez, Laura; Verdaguer i Espaulella, Xavier; Ribas de Pouplana, Lluis; Riera i Escalé, Antoni |
22-Oct-2021 | Recent Advances in the Enantioselective Synthesis of Chiral Amines via Transition Metal-Catalyzed Asymmetric Hydrogenation | Cabré, Albert; Verdaguer i Espaulella, Xavier; Riera i Escalé, Antoni |
25-Mar-2021 | Structure-based design of a Cortistatin analogue with immunomodulatory activity in models of inflammatory bowel disease | Rol Rúa, Álvaro; Todorovski, Toni; Martin-Malpartida, Pau; Escolà Jané, Anna; Gonzalez-Rey, Elena; Aragón Altarriba, Eric; Verdaguer i Espaulella, Xavier; Vallès Miret, Mariona; Farrera Sinfreu, Josep Maria; Puig, Eduard; Fernández-Carneado, Jimena; Ponsati, Berta; Delgado, Mario; Riera i Escalé, Antoni; Macías Hernández, María J. |
14-Feb-2023 | P-Stereogenic Ir-MaxPHOX: A Step toward Privileged Catalysts for Asymmetric Hydrogenation of Nonchelating Olefins | Biosca, Maria; Cruz Sánchez, Pol de la; Faiges, Jorge; Margalef, Jèssica; Salomó i Prat, Ernest; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier; Ferré, Joan; Maseras, Feliu; Besora, Maria; Pàmies, Oscar; Diéguez, Montserrat |
18-Jan-2023 | Synthesis and Biological Activity of a VHL-Based PROTAC Specific for p38α | Cubillos Rojas, Mónica; Loren, Guillem; Hakim, Yusuf Z.; Verdaguer i Espaulella, Xavier; Riera i Escalé, Antoni; Nebreda, Àngel R. |
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