Search


Current filters:

Start a new search
Add filters:

Use filters to refine the search results.


Results 1-10 of 10 (Search time: 0.027 seconds).
  • previous
  • 1
  • next
Item hits:
Issue DateTitleAuthor(s)
14-Sep-2022Design and optimization of oestrogen receptor PROTACs based on 4-hydroxytamoxifenLoren, Guillem; Espuny, Irene; Llorente Lope, Alicia; Donoghue, Craig; Verdaguer i Espaulella, Xavier; Gomis, Roger R.; Riera i Escalé, Antoni
11-May-2022Iridium-catalyzed asymmetric hydrogenation of 2,3-diarylallyl amines with a threonine-derived P-stereogenic ligand for the synthesis of tetrahydroquinolines and tetrahydroisoquinolinesRojo, Pep; Molinari, Medea; Cabré, Albert; García-Mateos, Clara; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
3-Jun-2021BOM-phosphinite as an electrophilic P-stereogenic transfer reagent for the synthesis of bulky phosphines. Synthesis of tert-butyl(3,5-di-tert-butylphenyl)BisP*Rojo, Pep; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
12-May-2022Amino acids with fluorescent tetrazine ethers as bioorthogonal handles for peptide modificationRos, Enric; Bellido, Marina; Matarin, Joan A.; Gallen, Albert; Martínez, Manuel; Rodríguez, Laura; Verdaguer i Espaulella, Xavier; Ribas de Pouplana, Lluis; Riera i Escalé, Antoni
11-Sep-2020Somatostatin, an in vivo binder to Aβ oligomers, Binds to βPFOAβ(1−42) TetramersPuig Gomà-Camps, Eduard; Tolchard, James; Riera i Escalé, Antoni; Carulla Casanovas, Natàlia
22-Oct-2021Recent Advances in the Enantioselective Synthesis of Chiral Amines via Transition Metal-Catalyzed Asymmetric HydrogenationCabré, Albert; Verdaguer i Espaulella, Xavier; Riera i Escalé, Antoni
25-Mar-2021Structure-based design of a Cortistatin analogue with immunomodulatory activity in models of inflammatory bowel diseaseRol Rúa, Álvaro; Todorovski, Toni; Martin-Malpartida, Pau; Escolà Jané, Anna; Gonzalez-Rey, Elena; Aragón Altarriba, Eric; Verdaguer i Espaulella, Xavier; Vallès Miret, Mariona; Farrera Sinfreu, Josep Maria; Puig, Eduard; Fernández-Carneado, Jimena; Ponsati, Berta; Delgado, Mario; Riera i Escalé, Antoni; Macías Hernández, María J.
14-Feb-2023P-Stereogenic Ir-MaxPHOX: A Step toward Privileged Catalysts for Asymmetric Hydrogenation of Nonchelating OlefinsBiosca, Maria; Cruz Sánchez, Pol de la; Faiges, Jorge; Margalef, Jèssica; Salomó i Prat, Ernest; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier; Ferré, Joan; Maseras, Feliu; Besora, Maria; Pàmies, Oscar; Diéguez, Montserrat
18-Jan-2023Synthesis and Biological Activity of a VHL-Based PROTAC Specific for p38αCubillos Rojas, Mónica; Loren, Guillem; Hakim, Yusuf Z.; Verdaguer i Espaulella, Xavier; Riera i Escalé, Antoni; Nebreda, Àngel R.
28-Dec-2023Discovery and Mechanistic Elucidation of NQO1-Bioactivatable Small Molecules That Overcome Resistance to Degraders.Barbosa, Bárbara M. G.; Sfyaki, Aikaterini; Rafael, Sergi; José-Duran, Ferran; Pous, Joan; Sánchez Zarzalejo, Carolina; Perez-Lopez, Carles; Vilanova, Mar; Cigler, Marko; Gay, Marina; Vilaseca, Marta; Winter, Georg E.; Riera i Escalé, Antoni; Mayor-Ruiz, Cristina