Browsing by Author Muñoz-Torrero López-Ibarra, Diego

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Issue DateTitleAuthor(s)
2018Development of hybrid compounds to tackle Alzheimer’s diseaseMuñoz-Torrero López-Ibarra, Diego; Pérez Areales, Francisco Javier
2022Discovery and In Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's DiseaseCodony Gisbert, Sandra; Pont Masanet, Caterina; Griñán Ferré, Christian; Di Pede-Mattatelli, Ania; Calvó-Tusell, Carla; Feixas, Ferran; Osuna, Sílvia; Jarné-Ferrer, Júlia; Naldi, Marina; Bartolini, Manuela; Loza, María Isabel; Brea, José; Bartolini; Pérez, Belén; Bartra, Clara; Sanfeliu i Pujol, Coral; Juárez Jiménez, Jordi; Morisseau, Christophe; Hammock, Bruce D.; Pallàs i Llibería, Mercè, 1964-; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego
2021Discovery of a Potent Dual Inhibitor of Acetylcholinesterase and Butyrylcholinesterase with Antioxidant Activity that Alleviates Alzheimer-like Pathology in Old APP/PS1 MiceViayna, Elisabet; Coquelle, Nicolas; Cieslikiewicz-Bouet, Monika; Cisternas, Pedro; Oliva, Carolina; Sánchez-López, E. (Elena); Ettcheto Arriola, Miren; Bartolini, Manuela; De Simone, Angela; Ricchini, Mattia; Rendina, Marisa; Pons, Mégane; Firuzi, Omidreza; Pérez, Belén; Saso, Luciano; Andrisano, Vincenza; Nachon, Florian; Brazzolotto, Xavier; García, Maria Luisa; Camins Espuny, Antoni; Silman, Israel; Jean, Ludovic; Inestrosa, Nibaldo C.; Colletier, Jacques-Philippe; Renard, Pierre-Yves; Muñoz-Torrero López-Ibarra, Diego
2022Discovery of Dual Aβ/Tau Inhibitors and Evaluation of Their Therapeutic Effect on a Drosophila Model of Alzheimer's DiseaseGandini, Annachiara; Gonçalves, Ana Elisa; Strocchi, Silvia; Albertini, Claudia; Janočková, Jana; Tramarin, Anna; Grifoni, Daniela; Poeta, Eleonora; Soukup, Ondrej; Muñoz-Torrero López-Ibarra, Diego; Monti, Barbara; Sabaté Lagunas, Raimon; Bartolini, Manuela; Legname, Giuseppe; Bolognesi, Maria Laura
22-Mar-2013Disseny i síntesi de nous compostos multipotents per al tractament de la malaltia d’AlzheimerViana Gaza, Maria Elisabet
4-May-2012Disseny, síntesi, avaluació farmacològica i modelatge molecular de nous inhibidors de l’acetilcolinesterasa de lloc d’unió dualGaldeano Cantador, Carlos
1-Aug-2013Dual inhibitors of beta-amyloid aggregation and acetylcholinesterase as multi-target anti-Alzheimer drug candidatesViayna, Elisabet; Sabaté Lagunas, Raimon; Muñoz-Torrero López-Ibarra, Diego
28-Oct-2020Evaluation of the effects of acetylcholinesterase inhibitors in the zebrafish touch-evoked response: quantitative vs. qualitative assessmentGuzman, Laura; Besa, Gisela; Linares, Daniela; González, Lara; Pont Masanet, Caterina; Bartolini, Manuela; Haigis, Ann-Cathrin; Legradi, Jessica; Muñoz-Torrero López-Ibarra, Diego; Gómez Catalán, Jesús; Barenys Espadaler, Marta
6-Nov-2015Exploring heterocyclic scaffolds in the development of multi-target anti-Alzheimer and multi-trypanosomatid compoundsDi Pietro, O.
16-Jan-2009La filtració al buitSeco, Miquel (Seco García); Casamitjana i Badia, Núria; Angurell Purroy, Inmaculada; Caubet Marín, Amparo; Dinarès Milà, M. Immaculada; Llor Brunés, Núria; Muñoz-Torrero López-Ibarra, Diego; Nicolás Galindo, Ernesto; Pérez García, M. Lluïsa (Maria Lluïsa); Pujol Dilmé, M. Dolors; Rosell Pellisé, Glòria; Velasco Castrillo, Dolores
23-Feb-2009La filtración a vacíoSeco, Miquel (Seco García); Casamitjana i Badia, Núria; Angurell Purroy, Inmaculada; Caubet Marín, Amparo; Dinarès Milà, M. Immaculada; Llor Brunés, Núria; Muñoz-Torrero López-Ibarra, Diego; Nicolás Galindo, Ernesto; Pérez García, M. Lluïsa (Maria Lluïsa); Pujol Dilmé, M. Dolors; Rosell Pellisé, Glòria; Velasco Castrillo, Dolores
2021From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effectsPont Masanet, Caterina; Ginex, Tiziana; Griñán Ferré, Christian; Scheiner, Matthias; Mattellone, Alexia; Martínez, Noemí; Arce, Elsa M.; Soriano-Fernández, Yolanda; Naldi, Marina; De Simone, Angela; Barenys Espadaler, Marta; Gómez Catalán, Jesús; Pérez, Belén; Sabaté Lagunas, Raimon; Andrisano, Vincenza; Loza, María Isabel; Brea, José; Bartolini, Manuela; Bolognesi, Maria Laura; Decker, Michael; Pallàs i Llibería, Mercè, 1964-; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
Apr-2013Human disease and drug pharmacology, complex as real lifeViayna, Elisabet; Sola, Irene; Di Pietro, O.; Muñoz-Torrero López-Ibarra, Diego
11-Mar-2018Increasing polarity in tacrine and huprine derivatives: Potent anticholinesterase agents for the treatment of myasthenia gravisGaldeano Cantador, Carlos; Coquelle, Nicolas; Cieslikiewicz-Bouet, Monika; Bartolini, Manuela; Pérez, Belén; Clos, Victòria; Silman, Israel; Jean, Ludovic; Colletier, Jacques-Philippe; Renard, Pierre-Yves; Muñoz-Torrero López-Ibarra, Diego
3-Apr-2015Interaction of prion protein with acetylcholinesterase: potential pathobiological implications in prion diseasesTorrent, Joan; Vílchez Acosta, Alba del Valle; Muñoz-Torrero López-Ibarra, Diego; Trovaslet, M.; Nachon, Florian; Chatonnet, A.; Grznarova, K.; Acquatella-Tran Van Ba, I.; Goffic, R. Le; Herzog, Laetitia; Béringue, V.; Rezaei, H.
13-Nov-2015Multicomponent-based synthesis and biological evaluation of tricyclic heterofused quinolines with multi-trypanosomatid activityDi Pietro, O.; Vicente García, Esther; Taylor, Martin C.; Berenguer, Diana; Viayna, Elisabet; Lanzoni, Anna; Sola, Irene; Sayago, Helena; Riera Lizandra, Ma. Cristina; Fisa Saladrigas, Roser; Clos, Victòria; Pérez Fernández, Belén; Kelly, John M.; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego
10-Mar-2015Multigram synthesis and in vivo efficacy studies of a novel multitarget anti-Alzheimer's compoundSola, Irene; Viayna, Elisabet; Gómez Nadal, Tània; Galdeano Cantador, Carlos; Cassina, Matteo; Camps García, Pelayo; Romeo, Margherita; Diomede, Luisa; Salmona, Mario; Franco, Pilar; Schaeffer, Mireille; Colantuono, Diego; Robin, David; Brunner, Daniela; Taub, Nicole; Hutter-Paier, Birgit; Muñoz-Torrero López-Ibarra, Diego
31-Jan-2020Multitarget strategies in search of novel drug candidates against Alzheimer’s diseasePont Masanet, Caterina
4-Sep-2018Neuroprotective effects of the multitarget agent AVCRI104P3 in brain of middle-aged miceRelat, Julia; Come, Julio; Perez, B.; Camps García, Pelayo; Muñoz-Torrero López-Ibarra, Diego; Badia, Albert; Giménez Llort, Lydia; Clos, Victòria
15-Nov-2016Novel approaches toward anti-Alzheimer and antiprotozoal drug candidatesSola, Irene