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Results 1-10 of 19 (Search time: 0.021 seconds).
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Issue DateTitleAuthor(s)
14-Aug-2019Synthesis, in vitro profiling, and in vivo efficacy studies of a new family of multitarget anti-Alzheimer compoundsPérez Areales, Francisco Javier; Garrido, María; Aso Pérez, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró Colomé, Alba; Ginex, Tiziana; Sabaté Lagunas, Raimon; Pérez, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Ferrer, Isidro (Ferrer Abizanda); Ciruela Alférez, Francisco; Messeguer i Peypoch, Àngel, 1946-; Muñoz-Torrero López-Ibarra, Diego
28-Dec-2019Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6Vanden Eynde, Jean Jacques; Mangoni, Arduino A.; Rautio, Jarkko; Leprince, Jérôme; Azuma, Yasu-Taka; García-Sosa, Alfonso T.; Hulme, Christopher; Jampilek, Josef; Karaman, Rafik; Li, Wei; Gomes, Paula A. C; Hadjipavlou-Litina, Dimitra; Capasso, Raffaele; Geronikaki, Athina; Cerchia, Laura; Sabatier, Jean-Marc; Ragno, Rino; Tuccinardi, Tiziano; Trabocchi, Andrea; Winum, Jean-Yves; Luque Garriga, F. Xavier; Prokai-Tatrai, Katalin; Spetea, Mariana; Gütschow, Michael; Kosalec, Ivan; Guillou, Catherine; Vasconcelos, M. Helena; Kokotos, George; Rastelli, Giulio; de Sousa, Maria Emília; Manera, Clementina; Gemma, Sandra; Mangani, Stefano; Siciliano, Carlo; Galdiero, Stefania; Liu, Hong; Scott, Peter J. H.; de los Ríos, Cristóbal; Agrofoglio, Luigi A.; Collina, Simona; Guedes, Rita C.; Muñoz-Torrero López-Ibarra, Diego
10-Mar-2015Multigram synthesis and in vivo efficacy studies of a novel multitarget anti-Alzheimer's compoundSola, Irene; Viayna, Elisabet; Gómez Nadal, Tània; Galdeano Cantador, Carlos; Cassina, Matteo; Camps García, Pelayo; Romeo, Margherita; Diomede, Luisa; Salmona, Mario; Franco, Pilar; Schaeffer, Mireille; Colantuono, Diego; Robin, David; Brunner, Daniela; Taub, Nicole; Hutter-Paier, Birgit; Muñoz-Torrero López-Ibarra, Diego
13-Nov-2015Multicomponent-based synthesis and biological evaluation of tricyclic heterofused quinolines with multi-trypanosomatid activityDi Pietro, O.; Vicente García, Esther; Taylor, Martin C.; Berenguer, Diana; Viayna, Elisabet; Lanzoni, Anna; Sola, Irene; Sayago, Helena; Riera Lizandra, Ma. Cristina; Fisa Saladrigas, Roser; Clos, Victòria; Pérez Fernández, Belén; Kelly, John M.; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego
1-Dec-2014Synthesis and antiprotozoal activity of oligomethylene- and p-phenylene-bis(methylene)-linked bis(+)-huprinesSola, Irene; Artigas, Albert; Taylor, Martin C.; Gbedema, Stephen Y.; Pérez Fernández, Belén; Clos, Victòria; Wright, Colin W.; Kelly, John M.; Muñoz-Torrero López-Ibarra, Diego
1-Oct-2014Shogaol-huprine hybrids: Dual antioxidant and anticholinesterase agents with beta-amyloid and tau anti-aggregating propertiesPérez Areales, Francisco Javier; Di Pietro, O.; Espargaró Colomé, Alba; Vallverdú i Queralt, Anna; Galdeano Cantador, Carlos; Ragusa, Ilaria M.; Viayna, Elisabet; Guillou, Catherine; Clos, Victòria; Pérez Fernández, Belén; Sabaté Lagunas, Raimon; Lamuela Raventós, Rosa Ma.; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
22-Mar-2016Ultra rapid in vivo screening for anti-Alzheimer anti-amyloid drugsEspargaró Colomé, Alba; Medina, Aina; Di Pietro, O.; Muñoz-Torrero López-Ibarra, Diego; Sabaté Lagunas, Raimon
12-Sep-2014Tetrahydrobenzo[h][1,6]naphthyridine-6-chlorotacrine hybrids as a new family of anti-Alzheimer agents targeting beta-amyloid, tau, and cholinesterase pathologiesDi Pietro, O.; Pérez Areales, Francisco Javier; Juárez-Jiménez, Jordi; Espargaró Colomé, Alba; Clos, Victòria; Pérez Fernández, Belén; Lavilla Grífols, Rodolfo; Sabaté Lagunas, Raimon; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
Mar-2014Thioflavin-S staining of bacterial inclusion bodies for the fast, simple, and inexpensive screening of amyloid aggregation inhibitorsPouplana, Sergi; Espargaró Colomé, Alba; Galdeano Cantador, Carlos; Viayna, Elisabet; Sola, Irene; Ventura, Salvador; Muñoz-Torrero López-Ibarra, Diego; Sabaté Lagunas, Raimon
27-Mar-2014Synthesis and multi-target biological profiling of a novel family of rhein derivatives as disease-modifying anti-Alzheimer agentsViayna, Elisabet; Sola, Irene; Bartolini, Manuela; De Simone, Angela; Tapia-Rojas, Cheril; Serrano, Felipe G.; Sabaté Lagunas, Raimon; Juárez-Jiménez, Jordi; Pérez Fernández, Belén; Luque Garriga, F. Xavier; Andrisano, Vincenza; Clos, Victòria; Inestrosa, Nibaldo C.; Muñoz-Torrero López-Ibarra, Diego