Browsing by Author Pérez, Belén

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Issue DateTitleAuthor(s)
22-Jun-2021A bicyclic α-iminophosphonate improves cognitive decline in 5xFAD murine model of neurodegenerationEscolano Mirón, Carmen; Abás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Callado, Luis F.; Pérez, Belén; Pérez Lozano, Pilar; Brea, José; Loza, María Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A; García-Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Díaz, C.; Pérez, J.; Ramos Guerra, Cristian; Vicente, Filipa; Molins i Grau, Elies; Pallàs i Llibería, Mercè, 1964-
2019A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptorsPérez Areales, Francisco Javier; Turcu, Andreea L.; Barniol-Xicota, Marta; Pont Masanet, Caterina; Pivetta, Deborah; Espargaró Colomé, Alba; Bartolini, Manuela; De Simone, Angela; Andrisano, Vincenza; Pérez, Belén; Sabaté Lagunas, Raimon; Sureda, Francesc X.; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego
5-Nov-2022Allopurinol blocks aortic aneurysm in a mouse model of Marfan syndrome via reducing aortic oxidative stressRodríguez Rovira, Isaac; Arce, Cristina; De Rycke, Karo; Pérez, Belén; Carretero, Aitor; Arbonés, Marc; Teixidó Tura, Gisela; Gómez-Cabrera Mari Carmen; Campuzano Uceda, María Victoria; Jiménez Altayó, Francesc; Egea Guri, Gustavo
2022An Imidazoline 2 Receptor Ligand Relaxes Mouse Aorta via Off-Target Mechanisms Resistant to AgingJiménez Altayó, Francesc; Cabrera, Anna; Bagan Polonio, Andrea; Giménez-Llort, Lydia; Ocón, Pilar; Pérez, Belén; Pallàs i Llibería, Mercè, 1964-; Escolano Mirón, Carmen
20-Nov-2018Behavioral and Cognitive Improvement Induced by Novel Imidazoline I2 Receptor Ligands in Female SAMP8 MiceGriñán Ferré, Christian; Vasilopoulou, Foteini; Abás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Sureda, Francesc X.; Pérez, Belén; Callado, Luis F.; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Escolano Mirón, Carmen; Pallàs i Llibería, Mercè, 1964-
22-Jun-2021Benzofuranyl-2-imidazoles as imidazoline I2 receptor ligands for Alzheimer's diseaseRodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Pallàs i Llibería, Mercè, 1964-; Brocos-Mosquera, Iria; Callado, Luis F.; Loza, María Isabel; Martínez, Antón L.; Brea, José; Pérez, Belén; Molins i Grau, Elies; Jonghe, Steven de; Daelemans, Dirk; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Hernández-Hernández, Elena; García-Fuster, M. Julia; García-Sevilla, Jesús A.; Escolano Mirón, Carmen
19-Mar-2020Bicyclic alfa-iminophosphonates as high affinity imidazoline I2 receptor ligands for Alzheimer's diseaseAbás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Pérez, Belén; Molins i Grau, Elies; Luque Garriga, F. Xavier; Pérez Lozano, Pilar; Jonghe, Steven de; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, María Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Pallàs i Llibería, Mercè, 1964-; Callado, Luis F.; Escolano Mirón, Carmen
2021Clock/Sleep-Dependent Learning and Memory in Male 3xTg-AD Mice at Advanced Disease Stages and Extrinsic Effects of Huprine X and the Novel Multitarget Agent AVCRI104P3Giménez Llort, Lydia; Santana-Santana, Mikel; Ratia, Míriam; Pérez, Belén; Camps García, Pelayo; Muñoz-Torrero López-Ibarra, Diego; Badía, A. (Albert); Clos, Victòria
29-Sep-2021CPEB alteration and aberrant transcriptome-polyadenylation lead to a treatable SLC19A3 deficiency in Huntington's diseasePicó, Sara; Parras, Alberto; Santos Galindo, María; Pose Utrilla Julia; Castro, Margarita; Fraga, Enrique; Hernández, Ivo H.; Elorza, Ainara; Anta, Héctor; Wang, Nan; Martí Sánchez, Laura; Belloc, Eulàlia; Garcia Esparcia, Patricia; Garrido, Juan J.; Ferrer, Isidro; Macías García, Daniel; Mir, Pablo; Artuch, Rafael; Pérez, Belén; Hernández, Félix; Navarro, Pilar; López Sendón, José Luis; Iglesias, Teresa; Yang, X. William; Méndez, Raúl; Lucas, José J.
5-Jun-2022Design, synthesis, and in vitro and in vivo characterization of new memantine analogs for Alzheimer's diseaseTurcu, Andreea L.; Companys Alemany, Júlia; Phillips, Matthew B.; Patel, Dhilon S.; Griñán Ferré, Christian; Loza, María Isabel; Brea, José; Pérez, Belén; Soto del Cerro, David; Sureda, Francesc X.; Kurnikova, Maria G.; Johnson, Jon W.; Pallàs i Llibería, Mercè, 1964-; Vázquez Cruz, Santiago
2022Discovery and In Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's DiseaseCodony Gisbert, Sandra; Pont Masanet, Caterina; Griñán Ferré, Christian; Di Pede-Mattatelli, Ania; Calvó-Tusell, Carla; Feixas, Ferran; Osuna, Sílvia; Jarné-Ferrer, Júlia; Naldi, Marina; Bartolini, Manuela; Loza, María Isabel; Brea, José; Bartolini; Pérez, Belén; Bartra, Clara; Sanfeliu i Pujol, Coral; Juárez Jiménez, Jordi; Morisseau, Christophe; Hammock, Bruce D.; Pallàs i Llibería, Mercè, 1964-; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego
2021Discovery of a Potent Dual Inhibitor of Acetylcholinesterase and Butyrylcholinesterase with Antioxidant Activity that Alleviates Alzheimer-like Pathology in Old APP/PS1 MiceViayna, Elisabet; Coquelle, Nicolas; Cieslikiewicz-Bouet, Monika; Cisternas, Pedro; Oliva, Carolina; Sánchez-López, E. (Elena); Ettcheto Arriola, Miren; Bartolini, Manuela; De Simone, Angela; Ricchini, Mattia; Rendina, Marisa; Pons, Mégane; Firuzi, Omidreza; Pérez, Belén; Saso, Luciano; Andrisano, Vincenza; Nachon, Florian; Brazzolotto, Xavier; García, Maria Luisa; Camins Espuny, Antoni; Silman, Israel; Jean, Ludovic; Inestrosa, Nibaldo C.; Colletier, Jacques-Philippe; Renard, Pierre-Yves; Muñoz-Torrero López-Ibarra, Diego
2021From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effectsPont Masanet, Caterina; Ginex, Tiziana; Griñán Ferré, Christian; Scheiner, Matthias; Mattellone, Alexia; Martínez, Noemí; Arce, Elsa M.; Soriano-Fernández, Yolanda; Naldi, Marina; De Simone, Angela; Barenys Espadaler, Marta; Gómez Catalán, Jesús; Pérez, Belén; Sabaté Lagunas, Raimon; Andrisano, Vincenza; Loza, María Isabel; Brea, José; Bartolini, Manuela; Bolognesi, Maria Laura; Decker, Michael; Pallàs i Llibería, Mercè, 1964-; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
11-Mar-2018Increasing polarity in tacrine and huprine derivatives: Potent anticholinesterase agents for the treatment of myasthenia gravisGaldeano Cantador, Carlos; Coquelle, Nicolas; Cieslikiewicz-Bouet, Monika; Bartolini, Manuela; Pérez, Belén; Clos, Victòria; Silman, Israel; Jean, Ludovic; Colletier, Jacques-Philippe; Renard, Pierre-Yves; Muñoz-Torrero López-Ibarra, Diego
12-May-2022Insights into the Pharmacokinetics and In Vitro Cell-Based Studies of the Imidazoline I2 Receptor Ligand B06Bagan Polonio, Andrea; Morales-García, José A.; Griñán Ferré, Christian; Díaz, Caridad; Pérez del Palacio, José; Ramos, Maria C.; Vicente, Francisca; Pérez, Belén; Brea, José; Loza, María Isabel; Pallàs i Llibería, Mercè, 1964-; Escolano Mirón, Carmen
2-Jun-2020Pharmacological Inhibition of Soluble Epoxide Hydrolase as a New Therapy for Alzheimer's DiseaseGriñán Ferré, Christian; Codony Gisbert, Sandra; Pujol Bech, Eugènia; Yang, Jun; Leiva Martínez, Rosana; Escolano Mirón, Carmen; Puigoriol Illamola, Dolors; Companys Alemany, Júlia; Corpas Expósito, Rubén; Sanfeliu i Pujol, Coral; Pérez, Belén; Loza, María Isabel; Brea, José; Morisseau, Christophe; Hammock, Bruce D.; Vázquez Cruz, Santiago; Pallàs i Llibería, Mercè, 1964-; Galdeano Cantador, Carlos
2020Pharmacology and preclinical validation of a novel anticancer compound targeting PEPCK-MAragó, Marc; Moreno Felici, Juan; Abás Prades, Sònia; Rodríguez Arévalo, Sergio; Hyrossová, Petra; Figueras, Agnes; Viñals Canals, Francesc; Pérez, Belén; Loza, María Isabel; Brea, José; Latorre, Pedro; Carrodeguas, Jose A.; García-Roves, Pablo M. (Pablo Miguel); Galdeano, Carlos; Ginex, Tiziana; Luque Garriga, F. Xavier; Escolano Mirón, Carmen; Perales Losa, Carlos
21-Jan-2020Stenosis coexists with compromised α1-adrenergic contractions in the ascending aorta of a mouse model of Williams-Beuren syndromeJiménez Altayó, Francesc; Ortiz Romero, Paula; Puertas Umbert, Lídia; Dantas, Ana Paula; Pérez, Belén; Vila, Elisabet; D'Ocon, Pilar; Campuzano Uceda, María Victoria
1-Dec-2022Structure-Based Virtual Screening and in vitro and in vivo Analyses Revealed Potent Methyltransferase G9a Inhibitors as Prospective Anti-Alzheimer's AgentsBellver-Sanchis, Aina; Bhanwar Singh Choudhary; Companys Alemany, Júlia; Sukanya; Ávila-López, Pedro A.; Martínez Rodríguez, Antón Leandro; Brea Floriani, Jose Manuel; Malik, Ruchi; Pallàs i Llibería, Mercè, 1964-; Pérez, Belén; Griñán Ferré, Christian
14-Aug-2019Synthesis, in vitro profiling, and in vivo efficacy studies of a new family of multitarget anti-Alzheimer compoundsPérez Areales, Francisco Javier; Garrido, María; Aso Pérez, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró Colomé, Alba; Ginex, Tiziana; Sabaté Lagunas, Raimon; Pérez, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Ferrer, Isidro (Ferrer Abizanda); Ciruela Alférez, Francisco; Messeguer i Peypoch, Àngel, 1946-; Muñoz-Torrero López-Ibarra, Diego