Browsing by Author Pérez, Belén

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Issue DateTitleAuthor(s)
5-Jun-2022Design, synthesis, and in vitro and in vivo characterization of new memantine analogs for Alzheimer's diseaseTurcu, Andreea L.; Companys Alemany, Júlia; Phillips, Matthew B.; Patel, Dhilon S.; Griñán Ferré, Christian; Loza, María Isabel; Brea, José; Pérez, Belén; Soto del Cerro, David; Sureda, Francesc X.; Kurnikova, Maria G.; Johnson, Jon W.; Pallàs i Llibería, Mercè, 1964-; Vázquez Cruz, Santiago
2022Discovery and In Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's DiseaseCodony Gisbert, Sandra; Pont Masanet, Caterina; Griñán Ferré, Christian; Di Pede-Mattatelli, Ania; Calvó-Tusell, Carla; Feixas, Ferran; Osuna, Sílvia; Jarné-Ferrer, Júlia; Naldi, Marina; Bartolini, Manuela; Loza, María Isabel; Brea, José; Bartolini; Pérez, Belén; Bartra, Clara; Sanfeliu i Pujol, Coral; Juárez Jiménez, Jordi; Morisseau, Christophe; Hammock, Bruce D.; Pallàs i Llibería, Mercè, 1964-; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego
2021Discovery of a Potent Dual Inhibitor of Acetylcholinesterase and Butyrylcholinesterase with Antioxidant Activity that Alleviates Alzheimer-like Pathology in Old APP/PS1 MiceViayna, Elisabet; Coquelle, Nicolas; Cieslikiewicz-Bouet, Monika; Cisternas, Pedro; Oliva, Carolina; Sánchez-López, E. (Elena); Ettcheto Arriola, Miren; Bartolini, Manuela; De Simone, Angela; Ricchini, Mattia; Rendina, Marisa; Pons, Mégane; Firuzi, Omidreza; Pérez, Belén; Saso, Luciano; Andrisano, Vincenza; Nachon, Florian; Brazzolotto, Xavier; García, Maria Luisa; Camins Espuny, Antoni; Silman, Israel; Jean, Ludovic; Inestrosa, Nibaldo C.; Colletier, Jacques-Philippe; Renard, Pierre-Yves; Muñoz-Torrero López-Ibarra, Diego
2021From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effectsPont Masanet, Caterina; Ginex, Tiziana; Griñán Ferré, Christian; Scheiner, Matthias; Mattellone, Alexia; Martínez, Noemí; Arce, Elsa M.; Soriano-Fernández, Yolanda; Naldi, Marina; De Simone, Angela; Barenys Espadaler, Marta; Gómez Catalán, Jesús; Pérez, Belén; Sabaté Lagunas, Raimon; Andrisano, Vincenza; Loza, María Isabel; Brea, José; Bartolini, Manuela; Bolognesi, Maria Laura; Decker, Michael; Pallàs i Llibería, Mercè, 1964-; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
11-Mar-2018Increasing polarity in tacrine and huprine derivatives: Potent anticholinesterase agents for the treatment of myasthenia gravisGaldeano Cantador, Carlos; Coquelle, Nicolas; Cieslikiewicz-Bouet, Monika; Bartolini, Manuela; Pérez, Belén; Clos, Victòria; Silman, Israel; Jean, Ludovic; Colletier, Jacques-Philippe; Renard, Pierre-Yves; Muñoz-Torrero López-Ibarra, Diego
12-May-2022Insights into the Pharmacokinetics and In Vitro Cell-Based Studies of the Imidazoline I2 Receptor Ligand B06Bagan Polonio, Andrea; Morales-García, José A.; Griñán Ferré, Christian; Díaz, Caridad; Pérez del Palacio, José; Ramos, Maria C.; Vicente, Francisca; Pérez, Belén; Brea, José; Loza, María Isabel; Pallàs i Llibería, Mercè, 1964-; Escolano Mirón, Carmen
2-Jun-2020Pharmacological Inhibition of Soluble Epoxide Hydrolase as a New Therapy for Alzheimer's DiseaseGriñán Ferré, Christian; Codony Gisbert, Sandra; Pujol Bech, Eugènia; Yang, Jun; Leiva Martínez, Rosana; Escolano Mirón, Carmen; Puigoriol Illamola, Dolors; Companys Alemany, Júlia; Corpas Expósito, Rubén; Sanfeliu i Pujol, Coral; Pérez, Belén; Loza, María Isabel; Brea, José; Morisseau, Christophe; Hammock, Bruce D.; Vázquez Cruz, Santiago; Pallàs i Llibería, Mercè, 1964-; Galdeano Cantador, Carlos
2020Pharmacology and preclinical validation of a novel anticancer compound targeting PEPCK-MAragó, Marc; Moreno Felici, Juan; Abás Prades, Sònia; Rodríguez Arévalo, Sergio; Hyrossová, Petra; Figueras, Agnes; Viñals Canals, Francesc; Pérez, Belén; Loza, María Isabel; Brea, José; Latorre, Pedro; Carrodeguas, Jose A.; García-Roves, Pablo M. (Pablo Miguel); Galdeano, Carlos; Ginex, Tiziana; Luque Garriga, F. Xavier; Escolano Mirón, Carmen; Perales Losa, Carlos
21-Jan-2020Stenosis coexists with compromised α1-adrenergic contractions in the ascending aorta of a mouse model of Williams-Beuren syndromeJiménez Altayó, Francesc; Ortiz Romero, Paula; Puertas Umbert, Lídia; Dantas, Ana Paula; Pérez, Belén; Vila, Elisabet; D'Ocon, Pilar; Campuzano Uceda, María Victoria
1-Dec-2022Structure-Based Virtual Screening and in vitro and in vivo Analyses Revealed Potent Methyltransferase G9a Inhibitors as Prospective Anti-Alzheimer's AgentsBellver-Sanchis, Aina; Bhanwar Singh Choudhary; Companys Alemany, Júlia; Sukanya; Ávila-López, Pedro A.; Martínez Rodríguez, Antón Leandro; Brea Floriani, Jose Manuel; Malik, Ruchi; Pallàs i Llibería, Mercè, 1964-; Pérez, Belén; Griñán Ferré, Christian
14-Aug-2019Synthesis, in vitro profiling, and in vivo efficacy studies of a new family of multitarget anti-Alzheimer compoundsPérez Areales, Francisco Javier; Garrido, María; Aso Pérez, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró Colomé, Alba; Ginex, Tiziana; Sabaté Lagunas, Raimon; Pérez, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Ferrer, Isidro (Ferrer Abizanda); Ciruela Alférez, Francisco; Messeguer i Peypoch, Àngel, 1946-; Muñoz-Torrero López-Ibarra, Diego
27-Oct-2022Synthesis, In Vitro Profiling, and In Vivo Evaluation of Benzohomoadamantane-Based Ureas for Visceral Pain: A New Indication for Soluble Epoxide Hydrolase InhibitorsCodony Gisbert, Sandra; Entrena, José M.; Calvó-Tusell, Carla; Jora, Beatrice Elena; González Cano, Rafael C.; Osuna, Sílvia; Corpas Expósito, Rubén; Morisseau, Christophe; Pérez, Belén; Barniol-Xicota, Marta; Griñán Ferré, Christian; Pérez, Concepción; Rodríguez-Franco, María Isabel; Martínez, Antón L.; Loza, María Isabel; Pallàs i Llibería, Mercè, 1964-; Verhelst, Steven H. L.; Sanfeliu i Pujol, Coral; Feixas, Ferran; Hammock, Bruce D.; Brea, José; Cobos, Enrique J.; Vázquez Cruz, Santiago
16-Jan-2018Tetrasubstituted imidazolium salts as potent antiparasitic agents against African and American trypanosomiasesGhashghaei, Ouldouz; Kielland, Nicola; Revés, Marc; Taylor, Martin C.; Kelly, John M.; Di Pietro, O.; Muñoz-Torrero López-Ibarra, Diego; Pérez, Belén; Lavilla Grífols, Rodolfo
24-Dec-2014Therapeutic strategies based on modified U1 snRNAs and chaperones for Sanfilippo C splicing mutationsMatos, Liliana; Canals Montferrer, Isaac; Dridi, Larbi; Choi, Yoo; Prata, Maria Joao; Jordan, Peter; Desviat, Lourdes R.; Pérez, Belén; Pshezhetsky, Alexey V.; Grinberg Vaisman, Daniel Raúl; Alves, Sandra; Vilageliu i Arqués, Lluïsa