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Issue Date | Title | Author(s) |
---|---|---|
14-Aug-2019 | Synthesis, in vitro profiling, and in vivo efficacy studies of a new family of multitarget anti-Alzheimer compounds | Pérez Areales, Francisco Javier; Garrido, María; Aso Pérez, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró Colomé, Alba; Ginex, Tiziana; Sabaté Lagunas, Raimon; Pérez, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Ferrer, Isidro (Ferrer Abizanda); Ciruela Alférez, Francisco; Messeguer i Peypoch, Àngel, 1946-; Muñoz-Torrero López-Ibarra, Diego |
12-Feb-2014 | 1,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: synthesis, pharmacological evaluation and mechanistic studies | Di Pietro, O.; Viayna, Elisabet; Vicente García, Esther; Bartolini, Manuela; Ramón, Rosario; Juárez-Jiménez, Jordi; Clos, Victòria; Pérez Fernández, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego |
27-Mar-2014 | Synthesis and multi-target biological profiling of a novel family of rhein derivatives as disease-modifying anti-Alzheimer agents | Viayna, Elisabet; Sola, Irene; Bartolini, Manuela; De Simone, Angela; Tapia-Rojas, Cheril; Serrano, Felipe G.; Sabaté Lagunas, Raimon; Juárez-Jiménez, Jordi; Pérez Fernández, Belén; Luque Garriga, F. Xavier; Andrisano, Vincenza; Clos, Victòria; Inestrosa, Nibaldo C.; Muñoz-Torrero López-Ibarra, Diego |
12-Sep-2014 | Tetrahydrobenzo[h][1,6]naphthyridine-6-chlorotacrine hybrids as a new family of anti-Alzheimer agents targeting beta-amyloid, tau, and cholinesterase pathologies | Di Pietro, O.; Pérez Areales, Francisco Javier; Juárez-Jiménez, Jordi; Espargaró Colomé, Alba; Clos, Victòria; Pérez Fernández, Belén; Lavilla Grífols, Rodolfo; Sabaté Lagunas, Raimon; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
1-Oct-2014 | Shogaol-huprine hybrids: Dual antioxidant and anticholinesterase agents with beta-amyloid and tau anti-aggregating properties | Pérez Areales, Francisco Javier; Di Pietro, O.; Espargaró Colomé, Alba; Vallverdú i Queralt, Anna; Galdeano Cantador, Carlos; Ragusa, Ilaria M.; Viayna, Elisabet; Guillou, Catherine; Clos, Victòria; Pérez Fernández, Belén; Sabaté Lagunas, Raimon; Lamuela Raventós, Rosa Ma.; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
1-Dec-2014 | Synthesis and antiprotozoal activity of oligomethylene- and p-phenylene-bis(methylene)-linked bis(+)-huprines | Sola, Irene; Artigas, Albert; Taylor, Martin C.; Gbedema, Stephen Y.; Pérez Fernández, Belén; Clos, Victòria; Wright, Colin W.; Kelly, John M.; Muñoz-Torrero López-Ibarra, Diego |
Mar-2014 | Thioflavin-S staining of bacterial inclusion bodies for the fast, simple, and inexpensive screening of amyloid aggregation inhibitors | Pouplana, Sergi; Espargaró Colomé, Alba; Galdeano Cantador, Carlos; Viayna, Elisabet; Sola, Irene; Ventura, Salvador; Muñoz-Torrero López-Ibarra, Diego; Sabaté Lagunas, Raimon |
13-Nov-2015 | Multicomponent-based synthesis and biological evaluation of tricyclic heterofused quinolines with multi-trypanosomatid activity | Di Pietro, O.; Vicente García, Esther; Taylor, Martin C.; Berenguer, Diana; Viayna, Elisabet; Lanzoni, Anna; Sola, Irene; Sayago, Helena; Riera Lizandra, Ma. Cristina; Fisa Saladrigas, Roser; Clos, Victòria; Pérez Fernández, Belén; Kelly, John M.; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego |
15-May-2017 | Unveiling a Novel Transient Druggable Pocket in BACE-1 through Molecular Simulations: Conformational Analysis and Binding Mode of Multisite Inhibitors | Di Pietro, O.; Juárez Jiménez, Jordi; Muñoz-Torrero López-Ibarra, Diego; Laughton, Charles A.; Luque Garriga, F. Xavier |
16-Jan-2018 | Tetrasubstituted imidazolium salts as potent antiparasitic agents against African and American trypanosomiases | Ghashghaei, Ouldouz; Kielland, Nicola; Revés, Marc; Taylor, Martin C.; Kelly, John M.; Di Pietro, O.; Muñoz-Torrero López-Ibarra, Diego; Pérez, Belén; Lavilla Grífols, Rodolfo |
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