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Results 11-20 of 20 (Search time: 0.033 seconds).
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Issue DateTitleAuthor(s)
2022Discovery and In Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's DiseaseCodony Gisbert, Sandra; Pont Masanet, Caterina; Griñán Ferré, Christian; Di Pede-Mattatelli, Ania; Calvó-Tusell, Carla; Feixas, Ferran; Osuna, Sílvia; Jarné-Ferrer, Júlia; Naldi, Marina; Bartolini, Manuela; Loza, María Isabel; Brea, José; Bartolini; Pérez, Belén; Bartra, Clara; Sanfeliu i Pujol, Coral; Juárez Jiménez, Jordi; Morisseau, Christophe; Hammock, Bruce D.; Pallàs i Llibería, Mercè, 1964-; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego
2022Unveiling the Multitarget Anti-Alzheimer Drug Discovery Landscape: A Bibliometric AnalysisSampietro Pifarre, Anna; Pérez Areales, Francisco Javier; Martínez, Paula; Arce, Elsa M.; Galdeano Cantador, Carlos; Muñoz-Torrero López-Ibarra, Diego
2019A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptorsPérez Areales, Francisco Javier; Turcu, Andreea L.; Barniol-Xicota, Marta; Pont Masanet, Caterina; Pivetta, Deborah; Espargaró Colomé, Alba; Bartolini, Manuela; De Simone, Angela; Andrisano, Vincenza; Pérez, Belén; Sabaté Lagunas, Raimon; Sureda, Francesc X.; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego
2022A Combined Chronic Low-Dose Soluble Epoxide Hydrolase and Acetylcholinesterase Pharmacological Inhibition Promotes Memory Reinstatement in Alzheimer's Disease Mice ModelsJarné-Ferrer, Júlia; Griñán Ferré, Christian; Bellver-Sanchis, Aina; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego; Pallàs i Llibería, Mercè, 1964-
2023A novel rhein-huprine hybrid ameliorates disease-modifying properties in preclinical mice model of Alzheimer's disease exacerbated with high fat dietEspinosa-Jiménez, Triana; Cano Fernández, Amanda; Sánchez-López, E. (Elena); Olloquequi, Jordi; Folch, Jaume; Bulló, Mònica; Verdaguer Cardona, Ester; Auladell i Costa, M. Carme; Pont Masanet, Caterina; Muñoz-Torrero López-Ibarra, Diego; Parcerisas, Antoni; Camins Espuny, Antoni; Ettcheto Arriola, Miren
28-Oct-2020Evaluation of the effects of acetylcholinesterase inhibitors in the zebrafish touch-evoked response: quantitative vs. qualitative assessmentGuzman, Laura; Besa, Gisela; Linares, Daniela; González, Lara; Pont Masanet, Caterina; Bartolini, Manuela; Haigis, Ann-Cathrin; Legradi, Jessica; Muñoz-Torrero López-Ibarra, Diego; Gómez Catalán, Jesús; Barenys Espadaler, Marta
2023A rhein-huprine hybrid protects erythrocyte membrane integrity against Alzheimer's disease related Abeta(1-42) peptideZambrano, Pablo; Jemiola-Rzeminska, Malgorzata; Muñoz-Torrero López-Ibarra, Diego; Suwalsky, Mario; Strzalka, Kazimierz
2022Discovery of Dual Aβ/Tau Inhibitors and Evaluation of Their Therapeutic Effect on a Drosophila Model of Alzheimer's DiseaseGandini, Annachiara; Gonçalves, Ana Elisa; Strocchi, Silvia; Albertini, Claudia; Janočková, Jana; Tramarin, Anna; Grifoni, Daniela; Poeta, Eleonora; Soukup, Ondrej; Muñoz-Torrero López-Ibarra, Diego; Monti, Barbara; Sabaté Lagunas, Raimon; Bartolini, Manuela; Legname, Giuseppe; Bolognesi, Maria Laura
2021Protective Role of a Donepezil-Huprine Hybrid against the β-Amyloid (1-42) Effect on Human ErythrocytesZambrano, Pablo; Suwalsky, Mario; Jemiola-Rzeminska, Malgorzata; Gallardo-Nelson, María José; Strzalka, Kazimierz; Muñoz-Torrero López-Ibarra, Diego
2021From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effectsPont Masanet, Caterina; Ginex, Tiziana; Griñán Ferré, Christian; Scheiner, Matthias; Mattellone, Alexia; Martínez, Noemí; Arce, Elsa M.; Soriano-Fernández, Yolanda; Naldi, Marina; De Simone, Angela; Barenys Espadaler, Marta; Gómez Catalán, Jesús; Pérez, Belén; Sabaté Lagunas, Raimon; Andrisano, Vincenza; Loza, María Isabel; Brea, José; Bartolini, Manuela; Bolognesi, Maria Laura; Decker, Michael; Pallàs i Llibería, Mercè, 1964-; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego