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Issue DateTitleAuthor(s)
20-Nov-2018Behavioral and Cognitive Improvement Induced by Novel Imidazoline I2 Receptor Ligands in Female SAMP8 MiceGriñán Ferré, Christian; Vasilopoulou, Foteini; Abás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Sureda, Francesc X.; Pérez, Belén; Callado, Luis F.; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Escolano Mirón, Carmen; Pallàs i Llibería, Mercè, 1964-
19-Mar-2020Bicyclic alfa-iminophosphonates as high affinity imidazoline I2 receptor ligands for Alzheimer's diseaseAbás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Pérez, Belén; Molins i Grau, Elies; Luque Garriga, F. Xavier; Pérez Lozano, Pilar; Jonghe, Steven de; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, María Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Pallàs i Llibería, Mercè, 1964-; Callado, Luis F.; Escolano Mirón, Carmen
2022Discovery and In Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's DiseaseCodony Gisbert, Sandra; Pont Masanet, Caterina; Griñán Ferré, Christian; Di Pede-Mattatelli, Ania; Calvó-Tusell, Carla; Feixas, Ferran; Osuna, Sílvia; Jarné-Ferrer, Júlia; Naldi, Marina; Bartolini, Manuela; Loza, María Isabel; Brea, José; Bartolini; Pérez, Belén; Bartra, Clara; Sanfeliu i Pujol, Coral; Juárez Jiménez, Jordi; Morisseau, Christophe; Hammock, Bruce D.; Pallàs i Llibería, Mercè, 1964-; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego
1-Dec-2022Structure-Based Virtual Screening and in vitro and in vivo Analyses Revealed Potent Methyltransferase G9a Inhibitors as Prospective Anti-Alzheimer's AgentsBellver-Sanchis, Aina; Bhanwar Singh Choudhary; Companys Alemany, Júlia; Sukanya; Ávila-López, Pedro A.; Martínez Rodríguez, Antón Leandro; Brea Floriani, Jose Manuel; Malik, Ruchi; Pallàs i Llibería, Mercè, 1964-; Pérez, Belén; Griñán Ferré, Christian
12-May-2022Insights into the Pharmacokinetics and In Vitro Cell-Based Studies of the Imidazoline I2 Receptor Ligand B06Bagan Polonio, Andrea; Morales-García, José A.; Griñán Ferré, Christian; Díaz, Caridad; Pérez del Palacio, José; Ramos, Maria C.; Vicente, Francisca; Pérez, Belén; Brea, José; Loza, María Isabel; Pallàs i Llibería, Mercè, 1964-; Escolano Mirón, Carmen
2-Jun-2020Pharmacological Inhibition of Soluble Epoxide Hydrolase as a New Therapy for Alzheimer's DiseaseGriñán Ferré, Christian; Codony Gisbert, Sandra; Pujol Bech, Eugènia; Yang, Jun; Leiva Martínez, Rosana; Escolano Mirón, Carmen; Puigoriol Illamola, Dolors; Companys Alemany, Júlia; Corpas Expósito, Rubén; Sanfeliu i Pujol, Coral; Pérez, Belén; Loza, María Isabel; Brea, José; Morisseau, Christophe; Hammock, Bruce D.; Vázquez Cruz, Santiago; Pallàs i Llibería, Mercè, 1964-; Galdeano Cantador, Carlos
22-Jun-2021A bicyclic α-iminophosphonate improves cognitive decline in 5xFAD murine model of neurodegenerationEscolano Mirón, Carmen; Abás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Callado, Luis F.; Pérez, Belén; Pérez Lozano, Pilar; Brea, José; Loza, María Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A; García-Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Díaz, C.; Pérez, J.; Ramos Guerra, Cristian; Vicente, Filipa; Molins i Grau, Elies; Pallàs i Llibería, Mercè, 1964-
27-Oct-2022Synthesis, In Vitro Profiling, and In Vivo Evaluation of Benzohomoadamantane-Based Ureas for Visceral Pain: A New Indication for Soluble Epoxide Hydrolase InhibitorsCodony Gisbert, Sandra; Entrena, José M.; Calvó-Tusell, Carla; Jora, Beatrice Elena; González Cano, Rafael C.; Osuna, Sílvia; Corpas Expósito, Rubén; Morisseau, Christophe; Pérez, Belén; Barniol-Xicota, Marta; Griñán Ferré, Christian; Pérez, Concepción; Rodríguez-Franco, María Isabel; Martínez, Antón L.; Loza, María Isabel; Pallàs i Llibería, Mercè, 1964-; Verhelst, Steven H. L.; Sanfeliu i Pujol, Coral; Feixas, Ferran; Hammock, Bruce D.; Brea, José; Cobos, Enrique J.; Vázquez Cruz, Santiago
22-Jun-2021Benzofuranyl-2-imidazoles as imidazoline I2 receptor ligands for Alzheimer's diseaseRodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Pallàs i Llibería, Mercè, 1964-; Brocos-Mosquera, Iria; Callado, Luis F.; Loza, María Isabel; Martínez, Antón L.; Brea, José; Pérez, Belén; Molins i Grau, Elies; Jonghe, Steven de; Daelemans, Dirk; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Hernández-Hernández, Elena; García-Fuster, M. Julia; García-Sevilla, Jesús A.; Escolano Mirón, Carmen
2021From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effectsPont Masanet, Caterina; Ginex, Tiziana; Griñán Ferré, Christian; Scheiner, Matthias; Mattellone, Alexia; Martínez, Noemí; Arce, Elsa M.; Soriano-Fernández, Yolanda; Naldi, Marina; De Simone, Angela; Barenys Espadaler, Marta; Gómez Catalán, Jesús; Pérez, Belén; Sabaté Lagunas, Raimon; Andrisano, Vincenza; Loza, María Isabel; Brea, José; Bartolini, Manuela; Bolognesi, Maria Laura; Decker, Michael; Pallàs i Llibería, Mercè, 1964-; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego