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Issue Date | Title | Author(s) |
---|---|---|
7-Dec-2020 | Pharmacophore Modeling and 3D-QSAR Study of Indole and Isatin Derivatives as Antiamyloidogenic Agents Targeting Alzheimer's Disease | Purgatorio, Rosario; Gambacorta, Nicola; Catto, Marco; de Candia, Modesto; Pisani, Leonardo; Espargaró Colomé, Alba; Sabaté Lagunas, Raimon; Cellamare, Saverio; Nicolotti, Orazio; Altomare, Cosimo D. |
14-Aug-2019 | Synthesis, in vitro profiling, and in vivo efficacy studies of a new family of multitarget anti-Alzheimer compounds | Pérez Areales, Francisco Javier; Garrido, María; Aso Pérez, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró Colomé, Alba; Ginex, Tiziana; Sabaté Lagunas, Raimon; Pérez, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Ferrer, Isidro (Ferrer Abizanda); Ciruela Alférez, Francisco; Messeguer i Peypoch, Àngel, 1946-; Muñoz-Torrero López-Ibarra, Diego |
2021 | From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effects | Pont Masanet, Caterina; Ginex, Tiziana; Griñán Ferré, Christian; Scheiner, Matthias; Mattellone, Alexia; Martínez, Noemí; Arce, Elsa M.; Soriano-Fernández, Yolanda; Naldi, Marina; De Simone, Angela; Barenys Espadaler, Marta; Gómez Catalán, Jesús; Pérez, Belén; Sabaté Lagunas, Raimon; Andrisano, Vincenza; Loza, María Isabel; Brea, José; Bartolini, Manuela; Bolognesi, Maria Laura; Decker, Michael; Pallàs i Llibería, Mercè, 1964-; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
1-Oct-2014 | Shogaol-huprine hybrids: Dual antioxidant and anticholinesterase agents with beta-amyloid and tau anti-aggregating properties | Pérez Areales, Francisco Javier; Di Pietro, O.; Espargaró Colomé, Alba; Vallverdú i Queralt, Anna; Galdeano Cantador, Carlos; Ragusa, Ilaria M.; Viayna, Elisabet; Guillou, Catherine; Clos, Victòria; Pérez Fernández, Belén; Sabaté Lagunas, Raimon; Lamuela Raventós, Rosa Ma.; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
22-Apr-2016 | Key Points for the Amyloid Infectivity and Prion Neuronal Invasion | Espargaró Colomé, Alba; Busquets i Viñas, Ma. Antonia; Estelrich i Latràs, Joan; Sabaté Lagunas, Raimon |
22-Mar-2016 | Ultra rapid in vivo screening for anti-Alzheimer anti-amyloid drugs | Espargaró Colomé, Alba; Medina, Aina; Di Pietro, O.; Muñoz-Torrero López-Ibarra, Diego; Sabaté Lagunas, Raimon |
12-Sep-2014 | Tetrahydrobenzo[h][1,6]naphthyridine-6-chlorotacrine hybrids as a new family of anti-Alzheimer agents targeting beta-amyloid, tau, and cholinesterase pathologies | Di Pietro, O.; Pérez Areales, Francisco Javier; Juárez-Jiménez, Jordi; Espargaró Colomé, Alba; Clos, Victòria; Pérez Fernández, Belén; Lavilla Grífols, Rodolfo; Sabaté Lagunas, Raimon; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
27-Mar-2014 | Synthesis and multi-target biological profiling of a novel family of rhein derivatives as disease-modifying anti-Alzheimer agents | Viayna, Elisabet; Sola, Irene; Bartolini, Manuela; De Simone, Angela; Tapia-Rojas, Cheril; Serrano, Felipe G.; Sabaté Lagunas, Raimon; Juárez-Jiménez, Jordi; Pérez Fernández, Belén; Luque Garriga, F. Xavier; Andrisano, Vincenza; Clos, Victòria; Inestrosa, Nibaldo C.; Muñoz-Torrero López-Ibarra, Diego |
3-May-2012 | Using bacterial inclusion bodies to screen for amyloid aggregation inhibitors | Villar Piqué, Anna; Espargaró Colomé, Alba; Sabaté Lagunas, Raimon; Groot, Natalia S. de; Ventura, Salvador |
30-Oct-2022 | Three to Tango: Inhibitory Effect of Quercetin and Apigenin on Acetylcholinesterase, Amyloid-β Aggregation and Acetylcholinesterase-Amyloid Interaction | Alvarez-Berbel, Irene; Espargaró Colomé, Alba; Viayna, Elisabet; Caballero Hernández, Ana Belén; Busquets i Viñas, Ma. Antonia; Gámez Enamorado, Patrick; Luque Garriga, F. Xavier; Sabaté Lagunas, Raimon |
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