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Issue DateTitleAuthor(s)
12-Feb-20141,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: synthesis, pharmacological evaluation and mechanistic studiesDi Pietro, O.; Viayna, Elisabet; Vicente García, Esther; Bartolini, Manuela; Ramón, Rosario; Juárez-Jiménez, Jordi; Clos, Victòria; Pérez Fernández, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego
20081,2-Diaryl(3-pyridyl)ethanone Oximes. Intermolecular Hydrogen Bonding Networks Revealed by X-ray DiffractionAlcalde Pais, Ma. Ermitas (María de las Ermitas); Mesquida Estévez, Ma. Neus; Alvarez-Rúa, Carmen; Cuberes, Rosa; Frigola Mas, Jordi; García-Granda, Santiago
23-Apr-20091,2-Dimethylindole-3-sulfonyl (MIS) as protecting group for the side chain of arginineIsidro Llobet, Albert; Latassa, Daniel; Giraud, Matthieu; Álvarez Domingo, Mercedes; Albericio Palomera, Fernando
Jun-202011B-HSD1 inhibition rescues cognitive disturbances after chronic mild stress in mice: target engagement determination through TAPS assayPuigoriol Illamola, Dolors; Companys Alemany, Júlia; Mole, D. J.; Homer, N.; Vázquez Cruz, Santiago; Griñán Ferré, Christian; Pallàs i Llibería, Mercè, 1964-
9-Aug-201911β-HSD1 Inhibition Rescues SAMP8 Cognitive Impairment Induced by Metabolic StressPuigoriol Illamola, Dolors; Leiva Martínez, Rosana; Vázquez Carrera, Manuel; Vázquez Cruz, Santiago; Griñán Ferré, Christian; Pallàs i Llibería, Mercè, 1964-
1-Dec-20212-(Piperidin-4-yl)acetamides as Potent Inhibitors of Soluble Epoxide Hydrolase with Anti-Inflammatory ActivityMartín López, Juan; Codony Gisbert, Sandra; Bartra, Clara; Morisseau, Christophe; Loza, María Isabel; Sanfeliu i Pujol, Coral; Hammock, Bruce D.; Brea, José; Vázquez Cruz, Santiago
3-Oct-20223,4-Methylenedioxy methamphetamine, synthetic cathinones and psychedelics: From recreational to novel psychotherapeutic drugsLópez Arnau, Raúl; Camarasa García, Jordi; Lí Carbó, Marcel; Nadal-Gratacós, Núria; Puigseslloses, Pol; Espinosa-Velasco, María; Urquizu, Edurne; Escubedo Rafa, Elena; Pubill Sánchez, David
1-Mar-20133,4-Methylenedioxy-methamphetamine induces in vivo regional up-regulation of central nicotinic receptors in rats and potentiates the regulatory effects of nicotine on these receptorsPubill Sánchez, David; Garcia Ratés, Sara; Camarasa García, Jordi; Escubedo Rafa, Elena
28-Jun-20143,4-Methylenedioxymethamphetamine enhances kainic acid convulsive susceptibilityAbad, Sonia; Junyent Herena, Fèlix; Auladell i Costa, M. Carme; Pubill Sánchez, David; Pallàs i Llibería, Mercè, 1964-; Camarasa García, Jordi; Escubedo Rafa, Elena; Camins Espuny, Antoni
10-May-201946, Paladio, Pd. Un metal precioso con gran interés industrial y versatilidad sintéticaSolé Arjó, Daniel
5-Feb-20197,8-Dihydroxyflavone blocks the development of behavioral sensitization to MDPV, but not to cocaine: Differential role of the BDNF-TrkB pathwayDuart Castells, Leticia; López Arnau, Raúl; Vizcaíno, Sonia; Camarasa García, Jordi; Pubill Sánchez, David; Escubedo Rafa, Elena
22-Jun-2021A bicyclic α-iminophosphonate improves cognitive decline in 5xFAD murine model of neurodegenerationEscolano Mirón, Carmen; Abás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Callado, Luis F.; Pérez, Belén; Pérez Lozano, Pilar; Brea, José; Loza, María Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A; García-Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Díaz, C.; Pérez, J.; Ramos Guerra, Cristian; Vicente, Filipa; Molins i Grau, Elies; Pallàs i Llibería, Mercè, 1964-
29-May-2015A bioinspired peptide scaffold with high antibiotic activity and low in vivo toxicityRabanal Anglada, Francesc; Grau Campistany, Ariadna; Vila Farrés, Xavier; González-Linares, J. (Javier); Borràs Suárez, Miquel; Vila Estapé, Jordi; Manresa Presas, Ma. Ángeles (María Ángeles); Cajal Visa, Yolanda
2008A Biomimetic Enantioselective Approach to the Decahydroquinoline Class of Dendrobatid AlkaloidsAmat Tusón, Mercedes; Griera Farres, Rosa; Fabregat, Robert; Molins i Grau, Elies; Bosch Cartes, Joan
2022A Combined Chronic Low-Dose Soluble Epoxide Hydrolase and Acetylcholinesterase Pharmacological Inhibition Promotes Memory Reinstatement in Alzheimer's Disease Mice ModelsJarne Ferrer, Júlia; Griñán Ferré, Christian; Bellver Sanchis, Aina,; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego; Pallàs i Llibería, Mercè, 1964-
12-Aug-2020A fluorogenic cyclic peptide for imaging and quantification of drug-induced apoptosisBarth, Nicole D.; Subirós Funosas, Ramon; Mendive Tapia, Lorena; Duffin, Rodger; Shields, Mario A.; Cartwright, Jennifer A.; Troeira Henriques, Sónia; Sot, Jesus; Goñi, Felix M.; Lavilla Grífols, Rodolfo; Marwick, John A.; Vermeren, Sonja; Rossi, Adriano G.; Egeblad, Mikala; Dransfield, Ian; Vendrell, Marc
Feb-2016A general method for the synthesis of enantiopure 1,5-amino alcoholsGuignard, Guillaume Michel Pablo; Llor Brunés, Núria; Urbina Teixidor, Aina; Bosch Cartes, Joan; Amat Tusón, Mercedes
12-Jul-2010A general methodology for the enantioselective synthesis of 1-substituted tetrahydroisoquinoline alkaloidsAmat Tusón, Mercedes; Elias, Viviane; Llor Brunés, Núria; Subrizi, Fabiana; Molins i Grau, Elies; Bosch Cartes, Joan
20-Feb-2009A General Synthetic Route to Enantiopure 5-Substituted cis-DecahydroquinolinesAmat Tusón, Mercedes; Fabregat, Robert; Griera Farres, Rosa; Bosch Cartes, Joan
18-May-2015A Joint experimental-computational comparative study of the Pd(0)-catalysed reactions of aryl iodides and aldehydes with N, O, and S tethersSolé Arjó, Daniel; Mariani, Francesco; Fernández Cadenas, Israel