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Issue Date | Title | Author(s) |
---|---|---|
12-Feb-2014 | 1,2,3,4-Tetrahydrobenzo[h][1,6]naphthyridines as a new family of potent peripheral-to-midgorge-site inhibitors of acetylcholinesterase: synthesis, pharmacological evaluation and mechanistic studies | Di Pietro, O.; Viayna, Elisabet; Vicente García, Esther; Bartolini, Manuela; Ramón, Rosario; Juárez-Jiménez, Jordi; Clos, Victòria; Pérez Fernández, Belén; Andrisano, Vincenza; Luque Garriga, F. Xavier; Lavilla Grífols, Rodolfo; Muñoz-Torrero López-Ibarra, Diego |
1-Aug-2013 | Dual inhibitors of beta-amyloid aggregation and acetylcholinesterase as multi-target anti-Alzheimer drug candidates | Viayna, Elisabet; Sabaté Lagunas, Raimon; Muñoz-Torrero López-Ibarra, Diego |
27-Mar-2014 | Synthesis and multi-target biological profiling of a novel family of rhein derivatives as disease-modifying anti-Alzheimer agents | Viayna, Elisabet; Sola, Irene; Bartolini, Manuela; De Simone, Angela; Tapia-Rojas, Cheril; Serrano, Felipe G.; Sabaté Lagunas, Raimon; Juárez-Jiménez, Jordi; Pérez Fernández, Belén; Luque Garriga, F. Xavier; Andrisano, Vincenza; Clos, Victòria; Inestrosa, Nibaldo C.; Muñoz-Torrero López-Ibarra, Diego |
1-Oct-2014 | Shogaol-huprine hybrids: Dual antioxidant and anticholinesterase agents with beta-amyloid and tau anti-aggregating properties | Pérez Areales, Francisco Javier; Di Pietro, O.; Espargaró Colomé, Alba; Vallverdú i Queralt, Anna; Galdeano Cantador, Carlos; Ragusa, Ilaria M.; Viayna, Elisabet; Guillou, Catherine; Clos, Victòria; Pérez Fernández, Belén; Sabaté Lagunas, Raimon; Lamuela Raventós, Rosa Ma.; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
12-Sep-2014 | Tetrahydrobenzo[h][1,6]naphthyridine-6-chlorotacrine hybrids as a new family of anti-Alzheimer agents targeting beta-amyloid, tau, and cholinesterase pathologies | Di Pietro, O.; Pérez Areales, Francisco Javier; Juárez-Jiménez, Jordi; Espargaró Colomé, Alba; Clos, Victòria; Pérez Fernández, Belén; Lavilla Grífols, Rodolfo; Sabaté Lagunas, Raimon; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego |
Mar-2014 | Thioflavin-S staining of bacterial inclusion bodies for the fast, simple, and inexpensive screening of amyloid aggregation inhibitors | Pouplana, Sergi; Espargaró Colomé, Alba; Galdeano Cantador, Carlos; Viayna, Elisabet; Sola, Irene; Ventura, Salvador; Muñoz-Torrero López-Ibarra, Diego; Sabaté Lagunas, Raimon |
10-Mar-2015 | Multigram synthesis and in vivo efficacy studies of a novel multitarget anti-Alzheimer's compound | Sola, Irene; Viayna, Elisabet; Gómez Nadal, Tània; Galdeano Cantador, Carlos; Cassina, Matteo; Camps García, Pelayo; Romeo, Margherita; Diomede, Luisa; Salmona, Mario; Franco, Pilar; Schaeffer, Mireille; Colantuono, Diego; Robin, David; Brunner, Daniela; Taub, Nicole; Hutter-Paier, Birgit; Muñoz-Torrero López-Ibarra, Diego |
22-Mar-2016 | Ultra rapid in vivo screening for anti-Alzheimer anti-amyloid drugs | Espargaró Colomé, Alba; Medina, Aina; Di Pietro, O.; Muñoz-Torrero López-Ibarra, Diego; Sabaté Lagunas, Raimon |
2018 | Development of hybrid compounds to tackle Alzheimer’s disease | Muñoz-Torrero López-Ibarra, Diego; Pérez Areales, Francisco Javier |
2019 | A novel class of multitarget anti-Alzheimer benzohomoadamantane‒chlorotacrine hybrids modulating cholinesterases and glutamate NMDA receptors | Pérez Areales, Francisco Javier; Turcu, Andreea L.; Barniol-Xicota, Marta; Pont Masanet, Caterina; Pivetta, Deborah; Espargaró Colomé, Alba; Bartolini, Manuela; De Simone, Angela; Andrisano, Vincenza; Pérez, Belén; Sabaté Lagunas, Raimon; Sureda, Francesc X.; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego |
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