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Issue DateTitleAuthor(s)
22-Jun-2021Disease-modifying treatment with I2 imidazoline receptor ligand LSL60101 in an Alzheimer's disease mouse model: A Comparative study with donepezilVasilopoulou, Foteini; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Escolano Mirón, Carmen; Griñán Ferré, Christian; Pallàs i Llibería, Mercè, 1964-
2020Pharmacology and preclinical validation of a novel anticancer compound targeting PEPCK-MAragó, Marc; Moreno Felici, Juan; Abás Prades, Sònia; Rodríguez Arévalo, Sergio; Hyrossová, Petra; Figueras, Agnes; Viñals Canals, Francesc; Pérez, Belén; Loza, María Isabel; Brea, José; Latorre, Pedro; Carrodeguas, Jose A.; García-Roves, Pablo M. (Pablo Miguel); Galdeano, Carlos; Ginex, Tiziana; Luque Garriga, F. Xavier; Escolano Mirón, Carmen; Perales Losa, Carlos
May-2022A New Family of Subnanomolar inhibitors of Soluble Epoxide Hydrolase The FASEB journal, 13 May 2022, 36, supplement 1Escolano Mirón, Carmen; Bagan Polonio, Andrea; Turcu, Andreea L.; Morisseau, Christophe; Loza, María Isabel; Brea, José; Bartra, Clara; Sanfeliu i Pujol, Coral; Hammock, Bruce D.; Vázquez Cruz, Santiago
26-Aug-2021Microarray Analysis Revealed Inflammatory Transcriptomic Changes after LSL60101 Treatment in 5XFAD Mice ModelVasilopoulou, Foteini; Escolano Mirón, Carmen; Pallàs i Llibería, Mercè, 1964-; Griñán Ferré, Christian
19-Mar-2020Bicyclic alfa-iminophosphonates as high affinity imidazoline I2 receptor ligands for Alzheimer's diseaseAbás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Pérez, Belén; Molins i Grau, Elies; Luque Garriga, F. Xavier; Pérez Lozano, Pilar; Jonghe, Steven de; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, María Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Pallàs i Llibería, Mercè, 1964-; Callado, Luis F.; Escolano Mirón, Carmen
22-May-2020Amelioration of BPSD-like phenotype and cognitive decline in SAMP8 mice model accompanied by molecular changes after treatment with I2-imidazoline receptor ligand MCR5Vasilopoulou, Foteini; Bagan Polonio, Andrea; Rodríguez-Arévalo, Sergio; Escolano Mirón, Carmen; Griñán Ferré, Christian; Pallàs i Llibería, Mercè, 1964-
12-May-2022Insights into the Pharmacokinetics and In Vitro Cell-Based Studies of the Imidazoline I2 Receptor Ligand B06Bagan Polonio, Andrea; Morales-García, José A.; Griñán Ferré, Christian; Díaz, Caridad; Pérez del Palacio, José; Ramos, Maria C.; Vicente, Francisca; Pérez, Belén; Brea, José; Loza, María Isabel; Pallàs i Llibería, Mercè, 1964-; Escolano Mirón, Carmen
2-Jun-2020Pharmacological Inhibition of Soluble Epoxide Hydrolase as a New Therapy for Alzheimer's DiseaseGriñán Ferré, Christian; Codony Gisbert, Sandra; Pujol Bech, Eugènia; Yang, Jun; Leiva Martínez, Rosana; Escolano Mirón, Carmen; Puigoriol Illamola, Dolors; Companys Alemany, Júlia; Corpas Expósito, Rubén; Sanfeliu i Pujol, Coral; Pérez, Belén; Loza, María Isabel; Brea, José; Morisseau, Christophe; Hammock, Bruce D.; Vázquez Cruz, Santiago; Pallàs i Llibería, Mercè, 1964-; Galdeano Cantador, Carlos
31-Oct-2020I2 imidazoline receptor modulation protects aged SAMP8 mice against cognitive decline by suppressing the calcineurin pathwayVasilopoulou, Foteini; Griñán Ferré, Christian; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Escolano Mirón, Carmen; Pallàs i Llibería, Mercè, 1964-
23-Jun-2022Heterocycle-Based Multicomponent Reactions in Drug Discovery: From Hit Finding to Rational DesignNadal Rodríguez, Pau; Ghashghaei, Ouldouz; Bagan Polonio, Andrea; Escolano Mirón, Carmen; Lavilla Grífols, Rodolfo