Browsing by Author Brea, José

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Showing results 1 to 16 of 16
Issue DateTitleAuthor(s)
1-Dec-20212-(Piperidin-4-yl)acetamides as Potent Inhibitors of Soluble Epoxide Hydrolase with Anti-Inflammatory ActivityMartín López, Juan; Codony Gisbert, Sandra; Bartra, Clara; Morisseau, Christophe; Loza, María Isabel; Sanfeliu i Pujol, Coral; Hammock, Bruce D.; Brea, José; Vázquez Cruz, Santiago
22-Jun-2021A bicyclic α-iminophosphonate improves cognitive decline in 5xFAD murine model of neurodegenerationEscolano Mirón, Carmen; Abás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Callado, Luis F.; Pérez, Belén; Pérez Lozano, Pilar; Brea, José; Loza, María Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A; García-Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Díaz, C.; Pérez, J.; Ramos Guerra, Cristian; Vicente, Filipa; Molins i Grau, Elies; Pallàs i Llibería, Mercè, 1964-
May-2022A New Family of Subnanomolar inhibitors of Soluble Epoxide Hydrolase The FASEB journal, 13 May 2022, 36, supplement 1Escolano Mirón, Carmen; Bagan Polonio, Andrea; Turcu, Andreea L.; Morisseau, Christophe; Loza, María Isabel; Brea, José; Bartra, Clara; Sanfeliu i Pujol, Coral; Hammock, Bruce D.; Vázquez Cruz, Santiago
22-Mar-2020A Novel NMDA Receptor Antagonist Protects against Cognitive Decline Presented by Senescent MiceCompanys Alemany, Júlia; Turcu, Andreea L.; Bellver-Sanchis, Aina; Loza, María Isabel; Brea, José; Canudas Teixidó, Anna-Maria; Leiva Martínez, Rosana; Vázquez Cruz, Santiago; Pallàs i Llibería, Mercè, 1964-; Griñán Ferré, Christian
13-Sep-2022Amantadine variant - aryl conjugates that inhibit multiple M2 mutant - amantadine resistant influenza a virusesTzitzoglaki, Christina; Hoffmann, Anja; Turcu, Andreea L.; Schmerer, Patrick; Ma, Chulong; Laros, George; Liolios, Christos; Brea, José; Wang, Jun; Vázquez Cruz, Santiago; Schmidtke, Michaela; Kolocouris, Antonios
22-Jun-2021Benzofuranyl-2-imidazoles as imidazoline I2 receptor ligands for Alzheimer's diseaseRodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Pallàs i Llibería, Mercè, 1964-; Brocos-Mosquera, Iria; Callado, Luis F.; Loza, María Isabel; Martínez, Antón L.; Brea, José; Pérez, Belén; Molins i Grau, Elies; Jonghe, Steven de; Daelemans, Dirk; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Hernández-Hernández, Elena; García-Fuster, M. Julia; García-Sevilla, Jesús A.; Escolano Mirón, Carmen
19-Mar-2020Bicyclic alfa-iminophosphonates as high affinity imidazoline I2 receptor ligands for Alzheimer's diseaseAbás Prades, Sònia; Rodríguez-Arévalo, Sergio; Bagan Polonio, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos-Mosquera, Iria; Muguruza, Carolina; Pérez, Belén; Molins i Grau, Elies; Luque Garriga, F. Xavier; Pérez Lozano, Pilar; Jonghe, Steven de; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, María Isabel; Hernández-Hernández, Elena; García-Sevilla, Jesús A.; García-Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Pallàs i Llibería, Mercè, 1964-; Callado, Luis F.; Escolano Mirón, Carmen
5-Jun-2022Design, synthesis, and in vitro and in vivo characterization of new memantine analogs for Alzheimer's diseaseTurcu, Andreea L.; Companys Alemany, Júlia; Phillips, Matthew B.; Patel, Dhilon S.; Griñán Ferré, Christian; Loza, María Isabel; Brea, José; Pérez, Belén; Soto del Cerro, David; Sureda, Francesc X.; Kurnikova, Maria G.; Johnson, Jon W.; Pallàs i Llibería, Mercè, 1964-; Vázquez Cruz, Santiago
2022Discovery and In Vivo Proof of Concept of a Highly Potent Dual Inhibitor of Soluble Epoxide Hydrolase and Acetylcholinesterase for the Treatment of Alzheimer's DiseaseCodony Gisbert, Sandra; Pont Masanet, Caterina; Griñán Ferré, Christian; Di Pede-Mattatelli, Ania; Calvó-Tusell, Carla; Feixas, Ferran; Osuna, Sílvia; Jarné-Ferrer, Júlia; Naldi, Marina; Bartolini, Manuela; Loza, María Isabel; Brea, José; Bartolini; Pérez, Belén; Bartra, Clara; Sanfeliu i Pujol, Coral; Juárez Jiménez, Jordi; Morisseau, Christophe; Hammock, Bruce D.; Pallàs i Llibería, Mercè, 1964-; Vázquez Cruz, Santiago; Muñoz-Torrero López-Ibarra, Diego
2021From virtual screening hits targeting a cryptic pocket in BACE-1 to a nontoxic brain permeable multitarget anti-Alzheimer lead with disease-modifying and cognition-enhancing effectsPont Masanet, Caterina; Ginex, Tiziana; Griñán Ferré, Christian; Scheiner, Matthias; Mattellone, Alexia; Martínez, Noemí; Arce, Elsa M.; Soriano-Fernández, Yolanda; Naldi, Marina; De Simone, Angela; Barenys Espadaler, Marta; Gómez Catalán, Jesús; Pérez, Belén; Sabaté Lagunas, Raimon; Andrisano, Vincenza; Loza, María Isabel; Brea, José; Bartolini, Manuela; Bolognesi, Maria Laura; Decker, Michael; Pallàs i Llibería, Mercè, 1964-; Luque Garriga, F. Xavier; Muñoz-Torrero López-Ibarra, Diego
21-Jan-2016High-affinity sequence-selective DNA binding by iridium(III) polypyridyl organometallopeptidesGamba, Ilaria; Salvadó, Iria; Brissos, Rosa F.; Gámez Enamorado, Patrick; Brea, José; Loza, María Isabel; Vázquez, M. Eugenio; Vázquez López, Miguel
12-May-2022Insights into the Pharmacokinetics and In Vitro Cell-Based Studies of the Imidazoline I2 Receptor Ligand B06Bagan Polonio, Andrea; Morales-García, José A.; Griñán Ferré, Christian; Díaz, Caridad; Pérez del Palacio, José; Ramos, Maria C.; Vicente, Francisca; Pérez, Belén; Brea, José; Loza, María Isabel; Pallàs i Llibería, Mercè, 1964-; Escolano Mirón, Carmen
2-Jun-2020Pharmacological Inhibition of Soluble Epoxide Hydrolase as a New Therapy for Alzheimer's DiseaseGriñán Ferré, Christian; Codony Gisbert, Sandra; Pujol Bech, Eugènia; Yang, Jun; Leiva Martínez, Rosana; Escolano Mirón, Carmen; Puigoriol Illamola, Dolors; Companys Alemany, Júlia; Corpas Expósito, Rubén; Sanfeliu i Pujol, Coral; Pérez, Belén; Loza, María Isabel; Brea, José; Morisseau, Christophe; Hammock, Bruce D.; Vázquez Cruz, Santiago; Pallàs i Llibería, Mercè, 1964-; Galdeano Cantador, Carlos
2020Pharmacology and preclinical validation of a novel anticancer compound targeting PEPCK-MAragó, Marc; Moreno Felici, Juan; Abás Prades, Sònia; Rodríguez Arévalo, Sergio; Hyrossová, Petra; Figueras, Agnes; Viñals Canals, Francesc; Pérez, Belén; Loza, María Isabel; Brea, José; Latorre, Pedro; Carrodeguas, Jose A.; García-Roves, Pablo M. (Pablo Miguel); Galdeano, Carlos; Ginex, Tiziana; Luque Garriga, F. Xavier; Escolano Mirón, Carmen; Perales Losa, Carlos
27-Mar-2023Synthesis and Testing of Analogs of the Tuberculosis Drug Candidate SQ109 against Bacteria and Protozoa: Identification of Lead Compounds against Mycobacterium abscessus and Malaria ParasitesStampolaki, Marianna; Malwal, Satish R.; Álvarez-Cabrera, Nadine; Gao, Zijun; Moniruzzaman, Mohammad; Babii, Svitlana O.; Naziris, Nikolaos; Rey-Cibati, André; Valladares-Delgado, Mariana; Turcu, Andreea L.; Baek, Kyung-Hwa; Phan, Trong-Nhat; Lee, Hyeryon; Alcaraz, Mattheo; Watson, Savannah; Van der Watt, Mariette; Coertzen, Dina; Efstathiou, Natasa; Chountoulesi, Maria; Shoen, Carolyn M.; Papanastasiou, Ioannis P.; Brea, José; Cynamon, Michael H.; Birkholtz, Lyn-Marié; Kremer, Laurent; Hwan No, Joo; Vázquez Cruz, Santiago; Benaim, Gustavo; Demetzos, Costas; Zgurskaya, Helen I.; Dick, Thomas; Oldfield, Eric; Kolocouris, Antonios
27-Oct-2022Synthesis, In Vitro Profiling, and In Vivo Evaluation of Benzohomoadamantane-Based Ureas for Visceral Pain: A New Indication for Soluble Epoxide Hydrolase InhibitorsCodony Gisbert, Sandra; Entrena, José M.; Calvó-Tusell, Carla; Jora, Beatrice Elena; González Cano, Rafael C.; Osuna, Sílvia; Corpas Expósito, Rubén; Morisseau, Christophe; Pérez, Belén; Barniol-Xicota, Marta; Griñán Ferré, Christian; Pérez, Concepción; Rodríguez-Franco, María Isabel; Martínez, Antón L.; Loza, María Isabel; Pallàs i Llibería, Mercè, 1964-; Verhelst, Steven H. L.; Sanfeliu i Pujol, Coral; Feixas, Ferran; Hammock, Bruce D.; Brea, José; Cobos, Enrique J.; Vázquez Cruz, Santiago