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Results 11-20 of 41 (Search time: 0.028 seconds).
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Issue DateTitleAuthor(s)
11-May-2022Iridium-catalyzed asymmetric hydrogenation of 2,3-diarylallyl amines with a threonine-derived P-stereogenic ligand for the synthesis of tetrahydroquinolines and tetrahydroisoquinolinesRojo, Pep; Molinari, Medea; Cabré Montesinos, Albert; García-Mateos, Clara; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
Feb-2012Fine-tuning the [Pi]-[Pi]. Aromatic interactions in peptides: somatostatin analogues containing mesityl alanineMartín-Gago, Pablo; Gomez-Caminals, Marc; Ramón, Rosario; Verdaguer i Espaulella, Xavier; Martin-Malpartida, Pau; Aragón Altarriba, Eric; Fernández-Carneado, Jimena; Ponsati, Berta; López-Ruiz, Pilar; Cortes, María Alicia; Colás, Begoña; Macías Hernández, María J.; Riera i Escalé, Antoni
25-Mar-2021Structure-based design of a Cortistatin analogue with immunomodulatory activity in models of inflammatory bowel diseaseRol Rúa, Álvaro; Todorovski, Toni; Martin-Malpartida, Pau; Escolà Jané, Anna; González-Rey, Elena; Aragón Altarriba, Eric; Verdaguer i Espaulella, Xavier; Vallès Miret, Mariona; Farrera Sinfreu, Josep Maria; Puig Gomà-Camps, Eduard; Fernández-Carneado, Jimena; Ponsati, Berta; Delgado, Mario; Riera i Escalé, Antoni; Macías Hernández, María J.
12-May-2022Amino acids with fluorescent tetrazine ethers as bioorthogonal handles for peptide modificationRos, Enric; Bellido, Marina; Matarin, Joan A.; Gallen Ortiz, Albert; Martínez López, Manuel, 1957-; Rodríguez Raurell, Laura; Verdaguer i Espaulella, Xavier; Ribas de Pouplana, Lluis; Riera i Escalé, Antoni
28-Dec-2023Discovery and Mechanistic Elucidation of NQO1-Bioactivatable Small Molecules That Overcome Resistance to Degraders.Barbosa, Bárbara M. G.; Sfyaki, Aikaterini; Rafael, Sergi; José-Duran, Ferran; Pous, Joan; Sánchez Zarzalejo, Carolina; Perez-Lopez, Carles; Vilanova, Mar; Cigler, Marko; Gay i Marín, Marina; Vilaseca Casas, Marta; Winter, Georg E.; Riera i Escalé, Antoni; Mayor-Ruiz, Cristina
22-Jun-2017Dialkylammonium tert-Butylmethylphosphinites: Stable Intermediates for the Synthesis of P-Stereogenic LigandsSalomó i Prat, Ernest; Prades, Amparo; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
30-Sep-2015Rhodium-Catalyzed Pauson−Khand Reaction Using a Small-Bite-Angle P‑Stereogenic C1‑Diphosphine LigandCristóbal Lecina, Edgar; Costantino, Andrea R.; Grabulosa, Arnald; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
29-Jun-2016EPI-001, a compound active against castration-resistant prostate cancer, targets transactivation unit 5 of the androgen receptorMol, Eva de; Fenwick, R. Bryn; Phang, Christopher T. W.; Buzón Redorta, Víctor; Szulc, Elzbieta Maria; Fuente Cebrián, Àlex de la; Escobedo Pascual, Albert; García Arroyo, Jesús; Bertoncini, Carlos W.; Estébanez Perpiñá, Eva; McEwan, Iain J.; Riera i Escalé, Antoni; Salvatella i Giralt, Xavier
17-May-2016Highly Enantioselective Iridium-Catalyzed Hydrogenation of Cyclic EnamidesSalomó i Prat, Ernest; Orgué Gassol, Sílvia; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
22-Mar-2016Efficient preparation of (S)- and (R)-tert-Butylmethylphosphine-Borane: a novel entry to important P-Stereogenic ligandsSalomó i Prat, Ernest; Orgué Gassol, Sílvia; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier