Carregant...
Miniatura

Tipus de document

Article

Versió

Versió publicada

Data de publicació

Llicència de publicació

cc-by (c) Juliachs Milà, Mercè et al., 2013
Si us plau utilitzeu sempre aquest identificador per citar o enllaçar aquest document: https://hdl.handle.net/2445/96264

Effectivity of pazopanib treatment in orthotopic models of human testicular germ cell tumors

Títol de la revista

Director/Tutor

ISSN de la revista

Títol del volum

Resum

Background: Cisplatin (CDDP) resistance in testicular germ cell tumors (GCTs) is still a clinical challenge, and one associated with poor prognosis. The purpose of this work was to test pazopanib, an anti-tumoral and anti-angiogenic multikinase inhibitor, and its combination with lapatinib (an anti-ErbB inhibitor) in mouse orthotopic models of human testicular GCTs. Methods: We used two different models of human testicular GCTs orthotopically grown in nude mice; a CDDP-sensitive choriocarcinoma (TGT38) and a new orthotopic model generated from a metastatic GCT refractory to first-line CDDP chemotherapy (TGT44). Nude mice implanted with these orthotopic tumors were treated with the inhibitors and the effect on tumoral growth and angiogenesis was evaluated. Results: TGT44 refractory tumor had an immunohistochemical profile similar to the original metastasis, with characteristics of yolk sac tumor. TGT44 did not respond when treated with cisplatin. In contrast, pazopanib had an anti-angiogenic effect and anti-tumor efficacy in this model. Pazopanib in combination with lapatinib in TGT38, an orthotopic model of choriocarcinoma had an additive effect blocking tumor growth. Conclusions: We present pazopanib as a possible agent for the alternative treatment of CDDP-sensitive and CDDP-refractory GCT patients, alone or in combination with anti-ErbB therapies.

Matèries (anglès)

Citació

Citació

JULIACHS MILÀ, Mercè, VIDAL-BEL, August, GARCÍA DEL MURO SOLANS, Xavier, PIULATS, Josep m., CONDOM I MUNDÓ, Enric, CASANOVAS I CASANOVAS, Oriol, GRAUPERA I GARCIA-MILÀ, Mariona, GERMÀ LLUCH, José ramón, VILLANUEVA GARATACHEA, Alberto, VIÑALS CANALS, Francesc. Effectivity of pazopanib treatment in orthotopic models of human testicular germ cell tumors. _BMC Cancer_. 2013. Vol. 13, núm. 382. [consulta: 23 de gener de 2026]. ISSN: 1471-2407. [Disponible a: https://hdl.handle.net/2445/96264]

Exportar metadades

JSON - METS

Compartir registre