Solid-Phase Synthesis of New Trp(Nps)-Containing Dipeptide Derivatives as TRPV1 Channel Blockers

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dc.contributor.authorPérez de Vega, M.J.
dc.contributor.authorGarcía-López, M.T.
dc.contributor.authorZaccaro, Laura
dc.contributor.authorRoyo Expósito, Miriam
dc.contributor.authorAlbericio Palomera, Fernando
dc.contributor.authorFernández-Carvajal, A.
dc.contributor.authorFerrer-Montiel, A.
dc.contributor.authorGonzález-Muñiz, R.
dc.date.accessioned2014-03-12T14:20:07Z
dc.date.available2014-03-12T14:20:07Z
dc.date.issued2010-07-15
dc.date.updated2014-03-12T14:20:07Z
dc.description.abstractTrp(Nps)-Lys-NH2 derivatives, bearing alkyl or guanidine groups either at the N-terminus or on the Lys side-chain or at both positions were conveniently prepared on solid-phase and evaluated as TRPV1 channel antagonists.
dc.format.extent10 p.
dc.format.mimetypeapplication/pdf
dc.identifier.idgrec613899
dc.identifier.issn1420-3049
dc.identifier.pmid20657400
dc.identifier.urihttps://hdl.handle.net/2445/51423
dc.language.isoeng
dc.publisherMDPI Publishing
dc.relation.isformatofReproducció del document publicat a: http://dx.doi.org/10.3390/molecules15074924
dc.relation.ispartofMolecules, 2010, vol. 15, num. 7, p. 4924-4933
dc.relation.urihttp://dx.doi.org/10.3390/molecules15074924
dc.rightscc-by (c) Pérez de Vega, M.J. et al., 2010
dc.rights.accessRightsinfo:eu-repo/semantics/openAccess
dc.rights.urihttp://creativecommons.org/licenses/by/3.0/es
dc.sourceArticles publicats en revistes (Química Inorgànica i Orgànica)
dc.subject.classificationSíntesi en fase sólida
dc.subject.classificationCanals iònics
dc.subject.classificationBioquímica
dc.subject.classificationAnalgèsics
dc.subject.classificationCiències de la salut
dc.subject.classificationProteïnes
dc.subject.classificationDianes farmacològiques
dc.subject.otherSolid-phase synthesis
dc.subject.otherIon channels
dc.subject.otherBiochemistry
dc.subject.otherAnalgesics
dc.subject.otherMedical sciences
dc.subject.otherProteins
dc.subject.otherDrug targeting
dc.titleSolid-Phase Synthesis of New Trp(Nps)-Containing Dipeptide Derivatives as TRPV1 Channel Blockers
dc.typeinfo:eu-repo/semantics/article
dc.typeinfo:eu-repo/semantics/publishedVersion

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