Browsing by Author Riera i Escalé, Antoni

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Issue DateTitleAuthor(s)
14-Sep-2022Design and optimization of oestrogen receptor PROTACs based on 4-hydroxytamoxifenLoren, Guillem; Espuny, Irene; Llorente Lope, Alicia; Donoghue, Craig; Verdaguer i Espaulella, Xavier; Gomis i Cabré, Roger; Riera i Escalé, Antoni
15-Sep-2023Design and Synthesis of Bifunctional Compounds for Targeted Protein Degradation and PhosphorylationLoren Parrondo, Guillem
23-Feb-2018Development of synthetic strategies for lasso peptides with anticancer activityMartín Gómez, Helena
22-Jun-2017Dialkylammonium tert-Butylmethylphosphinites: Stable Intermediates for the Synthesis of P-Stereogenic LigandsSalomó i Prat, Ernest; Prades, Amparo; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
26-Nov-2018Direct Asymmetric Hydrogenation of N-Methyl and N-Alkyl Imines with an Ir(III)H CatalystSalomó i Prat, Ernest; Gallen Ortiz, Albert; Sciortino, Giuseppe; Ujaque, Gregori; Grabulosa, Arnald; Lledós, Agustí (Lledós i Falcó); Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
28-Dec-2023Discovery and Mechanistic Elucidation of NQO1-Bioactivatable Small Molecules That Overcome Resistance to Degraders.Barbosa, Bárbara M. G.; Sfyaki, Aikaterini; Rafael, Sergi; José-Duran, Ferran; Pous, Joan; Sánchez Zarzalejo, Carolina; Perez-Lopez, Carles; Vilanova, Mar; Cigler, Marko; Gay i Marín, Marina; Vilaseca Casas, Marta; Winter, Georg E.; Riera i Escalé, Antoni; Mayor-Ruiz, Cristina
22-Mar-2016Efficient preparation of (S)- and (R)-tert-Butylmethylphosphine-Borane: a novel entry to important P-Stereogenic ligandsSalomó i Prat, Ernest; Orgué Gassol, Sílvia; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
5-Aug-2019Enantioselective Synthesis of β-Methyl Amines via Iridium-Catalyzed Asymmetric Hydrogenation of N-Sulfonyl Allyl Amines.Cabré Montesinos, Albert; Verdaguer i Espaulella, Xavier; Riera i Escalé, Antoni
29-Jun-2016EPI-001, a compound active against castration-resistant prostate cancer, targets transactivation unit 5 of the androgen receptorMol, Eva de; Fenwick, R. Bryn; Phang, Christopher T. W.; Buzón Redorta, Víctor; Szulc, Elzbieta Maria; Fuente Cebrián, Àlex de la; Escobedo Pascual, Albert; García Arroyo, Jesús; Bertoncini, Carlos W.; Estébanez Perpiñá, Eva; McEwan, Iain J.; Riera i Escalé, Antoni; Salvatella i Giralt, Xavier
27-Apr-2017Ethylene glycol assisted intermolecular Pauson-Khand reactionCabré Montesinos, Albert; Verdaguer i Espaulella, Xavier; Riera i Escalé, Antoni
16-Jan-2019Extending the substrate scope in the hydrogenation of unfunctionalized tetrasubstituted olefins with Ir-P stereogenic aminophosphine-oxazoline catalystsBiosca, Maria; Salomó i Prat, Ernest; Cruz Sánchez, Pol de la; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier; Pàmies, Oscar; Diéguez, Montserrat
Feb-2012Fine-tuning the [Pi]-[Pi]. Aromatic interactions in peptides: somatostatin analogues containing mesityl alanineMartín-Gago, Pablo; Gomez-Caminals, Marc; Ramón, Rosario; Verdaguer i Espaulella, Xavier; Martin-Malpartida, Pau; Aragón Altarriba, Eric; Fernández-Carneado, Jimena; Ponsati, Berta; López-Ruiz, Pilar; Cortes, María Alicia; Colás, Begoña; Macías Hernández, María J.; Riera i Escalé, Antoni
8-Nov-2019Highly enantioselective iridium-catalyzed hydrogenation of 2-aryl allyl phthalimidesCabré Montesinos, Albert; Romagnoli, Elia; Martínez-Balart, Pol; Verdaguer i Espaulella, Xavier; Riera i Escalé, Antoni
17-May-2016Highly Enantioselective Iridium-Catalyzed Hydrogenation of Cyclic EnamidesSalomó i Prat, Ernest; Orgué Gassol, Sílvia; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
5-May-2014Immunostaining Protocol: P-Smad2 (Xenograft and Mice)Calon, Alexandre; Espinet, Elisa; Palomo Ponce, Sergio; Tauriello, Daniele V. F.; Iglesias, Mar; Céspedes, María; Sevillano, Marta; Nadal, Cristina; Jung, Peter; Zhang, Xiang; Byrom, Daniel; Riera i Escalé, Antoni; Rossell, David; Mangues, Ramon; Massagué i Solé, Joan, 1953-; Sancho, Elena; Batlle, Eduard
5-Mar-2014Immunostaining Protocol: P-Stat3 (Xenograft and Mice)Calon, Alexandre; Espinet, Elisa; Palomo Ponce, Sergio; Tauriello, Daniele V. F.; Iglesias, Mar; Cespedes, María Virtudes; Sevillano, Marta; Nadal, Cristina; Jung, Peter; Zhang, Xiang H. F.; Byrom, Daniel; Riera i Escalé, Antoni; Rossell, David; Mangues, Ramon; Massagué i Solé, Joan, 1953-; Sancho, Elena; Batlle, Eduard
25-Nov-2013Insights into Structure-Activity Relationships of Somatostatin Analogs Containing Mesitylalanine.Martín-Gago, Pablo; Aragón Altarriba, Eric; Gomez-Caminals, Marc; Fernández-Carneado, Jimena; Ramón, Rosario; Martin-Malpartida, Pau; Verdaguer i Espaulella, Xavier; López-Ruiz, Pilar; Colás, Begoña; Cortes, María Alicia; Ponsati, Berta; Macías Hernández, María J.; Riera i Escalé, Antoni
11-Mar-2016Intermolecular Pauson-Khad reaction: study of the regioselectivity, photochemistry of the adducts and synthetic applicationsKhaizourane, Héléa
16-Apr-2019Iridium complexes with P-stereogenic phosphino imidazole ligands: Synthesis, structure and catalysisÁlvarez Yebra, Rubén; Rojo, Pep; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier
11-May-2022Iridium-catalyzed asymmetric hydrogenation of 2,3-diarylallyl amines with a threonine-derived P-stereogenic ligand for the synthesis of tetrahydroquinolines and tetrahydroisoquinolinesRojo, Pep; Molinari, Medea; Cabré Montesinos, Albert; García-Mateos, Clara; Riera i Escalé, Antoni; Verdaguer i Espaulella, Xavier